SCHEMBL8464669

SCHEMBL8464669

Cc1cc(Cl)ccc1N1N=C(C(=O)N2CCN(C)CC2)CC1c1ccc(Cl)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 3/20 0.48
CNR2 P34972 3/20 0.48
GABRA2 P47869 1/20 0.45
GABRB2 P47870 1/20 0.45
POLB P06746 1/20 0.44
LMNA P02545 1/20 0.44
TP53 P04637 1/20 0.44
ALOX15 P16050 1/20 0.44
TSHR P16473 1/20 0.44
AKR1C3 P42330 1/20 0.42
PDE5A O76074 4/20 0.41
PDE2A O00408 1/20 0.41
PDE11A Q9HCR9 1/20 0.41
PDE10A Q9Y233 1/20 0.41
KMT2A Q03164 1/20 0.41
HRH4 Q9H3N8 5/20 0.40
HRH3 Q9Y5N1 2/20 0.40
HRH1 P35367 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2016965 0.91 CNR1 (0.59) CNR1CNR2GABRA2GABRB2POLB
Hydrochloric Acid SCHEMBL2020512 0.90 CNR1 (0.58) CNR1CNR2GABRA2GABRB2POLB
SCHEMBL8470259 0.88 CNR1 (0.54) CNR1CNR2GABRA2GABRB2POLB
SCHEMBL12527317 0.83 CNR1 (0.52) CNR1CNR2LMNAPDE5A
SCHEMBL4598704 0.81 CNR1 (0.60) CNR1CNR2GABRA2GABRB2LMNA
SCHEMBL2015954 0.81 CNR2 (0.62) CNR1CNR2GABRA2GABRB2LMNA
SCHEMBL8464834 0.81 CNR1 (0.49) CNR1CNR2AKR1C3PDE5A
SCHEMBL2018944 0.80 CNR1 (0.55) CNR1CNR2POLBLMNATP53
SCHEMBL4607380 0.80 CNR1 (0.61) CNR1CNR2TSHRKMT2A
SCHEMBL2288238 0.80 CNR1 (0.61) CNR1CNR2TSHRKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1946777-A1 Substituted pyrazoline for preventing weight gain Laboratorios del Dr. Esteve S.A. (ES) 2008-07-23 EP disclosed