SCHEMBL8465769

SCHEMBL8465769

COc1ccc(-c2ccc(OC(=O)NN)cc2)cc1OC1CCCC1

nearest known ligand 0.67

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 14/20 0.67
PDE4B Q07343 14/20 0.67
PDE4D Q08499 14/20 0.67
PDE4C Q08493 13/20 0.67
POLB P06746 1/20 0.53
MAPK14 Q16539 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8464657 0.88 PDE4B (0.73) PDE4APDE4BPDE4DPDE4CPOLB
SCHEMBL7447872 0.83 PDE4B (0.77) PDE4APDE4BPDE4DPDE4CPOLB
SCHEMBL7440108 0.80 PDE4B (1.00) PDE4APDE4BPDE4DPDE4CPOLB
SCHEMBL8465041 0.80 PDE4A (0.71) PDE4APDE4BPDE4DPDE4CPOLB
SCHEMBL5823060 0.79 PDE4A (0.77) PDE4APDE4BPDE4DPDE4CPOLB
SCHEMBL8461881 0.79 PDE4A (0.79) PDE4APDE4BPDE4DPDE4CPOLB
SCHEMBL8465957 0.78 PDE4D (0.75) PDE4APDE4BPDE4DPDE4C
SCHEMBL7444846 0.78 PDE4A (1.00) PDE4APDE4BPDE4DPDE4CPOLB
SCHEMBL8885266 0.78 PDE4B (0.81) PDE4APDE4BPDE4DPDE4CPOLB
SCHEMBL8466532 0.78 PDE4D (0.67) PDE4APDE4BPDE4DPDE4CPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0745063-B1 SUBSTITUTED BIPHENYL DERIVATIVES AS PHOSPHODIESTERASE INHIBITORS AMERICAN HOME PROD (US) 1999-03-24 EP claimed