SCHEMBL8467739

SCHEMBL8467739

c1cc2sc(SSc3cc4cnccc4s3)cc2cn1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 6/20 0.53
TGFBR1 P36897 8/20 0.37
CHEK1 O14757 1/20 0.35
AURKA O14965 1/20 0.35
DAPK3 O43293 1/20 0.35
PRKD3 O94806 1/20 0.35
MAP4K4 O95819 1/20 0.35
PAK4 O96013 1/20 0.35
ABL1 P00519 1/20 0.35
RET P07949 1/20 0.35
PIM1 P11309 1/20 0.35
FGFR1 P11362 1/20 0.35
PRKACA P17612 1/20 0.35
FLT1 P17948 1/20 0.35
LTK P29376 1/20 0.35
GRK5 P34947 1/20 0.35
KDR P35968 1/20 0.35
MAPK8 P45983 1/20 0.35
CSNK1A1 P48729 1/20 0.35
CDK8 P49336 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26800749 0.85 CYP2A6 (0.50) CYP2A6TGFBR1CHEK1AURKADAPK3
SCHEMBL11071527 0.75 CYP2A6 (0.56) CYP2A6TGFBR1CHEK1AURKADAPK3
SCHEMBL7113297 0.73 CYP2A6 (0.55) CYP2A6TGFBR1CHEK1AURKADAPK3
SCHEMBL16023619 0.73 CYP2A6 (0.55) CYP2A6TGFBR1CHEK1AURKADAPK3
SCHEMBL11070896 0.73 CYP2A6 (0.65) CYP2A6TGFBR1CHEK1AURKADAPK3
SCHEMBL3483101 0.73 CYP2A6 (0.55) CYP2A6TGFBR1CHEK1AURKADAPK3
SCHEMBL10677527 0.73 CYP2A6 (0.55) CYP2A6TGFBR1CHEK1AURKADAPK3
SCHEMBL11643448 0.73 CYP2A6 (0.55) CYP2A6TGFBR1CHEK1AURKADAPK3
Hydrochloric Acid SCHEMBL27139693 0.72 CYP2A6 (0.62) CYP2A6TGFBR1CHEK1AURKADAPK3
SCHEMBL12689590 0.71 CYP2A6 (0.51) CYP2A6TGFBR1CHEK1AURKADAPK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5869591-A ELASTOMER COMPRISING CROSSLINKED PSEUDORANDOM INTERPOLYMER OF ALPHA-OLEFIN, VINYLIDENE AROMATIC COMPOUND, OPTIONAL DIENE THE DOW CHEMICAL COMPANY (US) 1999-02-09 US disclosed
US-4582539-A ADDING ZINC MODIFIED SILICA DERIVED FROM ALKALI METAL SILICATE AND ZINC SALT PHILLIPS PETROLEUM COMPANY (US) 1986-04-15 US disclosed
US-4390648-A ZINC MODIFIED SILICA, HYSTERESIS PHILLIPS PETROLEUM COMPANY (US) 1983-06-28 US disclosed