SCHEMBL8467911

SCHEMBL8467911

COc1ccc2c(c1)CCNC2.COc1ccc2c(c1)CCNC2

nearest known ligand 0.86

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CD274 Q9NZQ7 2/20 0.59
HTR2C P28335 2/20 0.57
HTR2A P28223 1/20 0.57
HTR2B P41595 1/20 0.57
KCNH2 Q12809 1/20 0.57
RYR2 Q92736 1/20 0.57
ASIC3 Q9UHC3 1/20 0.55
DRD2 P14416 2/20 0.51
DRD3 P35462 2/20 0.51
HRH3 Q9Y5N1 1/20 0.50
DRD1 P21728 1/20 0.50
DRD5 P21918 1/20 0.50
ADRA2A P08913 1/20 0.49
ADRA2B P18089 1/20 0.49
ADRA2C P18825 1/20 0.49
HTR7 P34969 1/20 0.49
NISCH Q9Y2I1 1/20 0.49
LMNA P02545 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP2D6 P10635 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL532484 1.00 CD274 (0.59) CD274HTR2CHTR2AHTR2BKCNH2
Hydrochloric Acid SCHEMBL587493 0.98 CD274 (0.58) CD274HTR2CHTR2AHTR2BKCNH2
SCHEMBL29558442 0.93 HTR2C (0.57) CD274HTR2CHTR2AHTR2BKCNH2
SCHEMBL746109 0.93 HTR2C (0.57) CD274HTR2CHTR2AHTR2BKCNH2
Hydrochloric Acid SCHEMBL1124555 0.91 HTR2C (0.55) CD274HTR2CHTR2AHTR2BKCNH2
Hydrochloric Acid SCHEMBL31062521 0.91 HTR2C (0.55) CD274HTR2CHTR2AHTR2BKCNH2
Oxalic Acid SCHEMBL7199943 0.91 CD274 (0.52) CD274HTR2CHTR2AHTR2BKCNH2
SCHEMBL29758918 0.89 KCNH2 (0.54) CD274HTR2CHTR2AHTR2BKCNH2
SCHEMBL4859823 0.89 KCNH2 (0.54) CD274HTR2CHTR2AHTR2BKCNH2
Bromide SCHEMBL19644475 0.89 CD274 (0.51) CD274HTR2CHTR2AHTR2BKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0869787-A4 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 1999-03-24 EP disclosed
EP-0869787-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1998-10-14 EP disclosed
WO-1997024119-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1997-07-10 WO disclosed