SCHEMBL8469552

SCHEMBL8469552

c1ccc2c(c1)CCCN2c1ccncn1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 2/20 0.63
NUDT1 P36639 1/20 0.47
MKNK1 Q9BUB5 3/20 0.44
MKNK2 Q9HBH9 3/20 0.44
L3MBTL1 Q9Y468 1/20 0.43
JAK2 O60674 2/20 0.42
JAK3 P52333 1/20 0.42
PTK2 Q05397 1/20 0.42
RXRA P19793 1/20 0.41
RXRB P28702 1/20 0.41
RXRG P48443 1/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
SIGMAR1 Q99720 1/20 0.41
MAPK8 P45983 1/20 0.40
MAPK9 P45984 1/20 0.40
POLB P06746 1/20 0.40
HSD17B10 Q99714 1/20 0.40
CYP2C9 P11712 1/20 0.39
IDO1 P14902 1/20 0.39
KCNH2 Q12809 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9379977 0.91 ROCK1 (0.61) ROCK1MKNK1MKNK2SMN1; SMN2MAPK8
SCHEMBL28609745 0.89 ROCK1 (0.60) ROCK1MKNK1MKNK2SMN1; SMN2MAPK8
SCHEMBL18012073 0.83 ROCK1 (0.64) ROCK1NUDT1L3MBTL1JAK2JAK3
SCHEMBL5245431 0.79 ROCK1 (0.63) ROCK1NUDT1L3MBTL1JAK2JAK3
SCHEMBL16071242 0.78 ROCK1 (0.58) ROCK1NUDT1L3MBTL1JAK2JAK3
SCHEMBL12968733 0.78 ROCK1 (1.00) ROCK1NUDT1MKNK1MKNK2MAPK8
SCHEMBL28667775 0.77 ROCK1 (0.53) ROCK1NUDT1L3MBTL1JAK2JAK3
SCHEMBL30362762 0.77 ROCK1 (0.53) ROCK1NUDT1L3MBTL1JAK2JAK3
SCHEMBL6761496 0.77 ROCK1 (0.72) ROCK1NUDT1MKNK1MKNK2L3MBTL1
SCHEMBL17033290 0.75 ROCK1 (0.62) ROCK1NUDT1L3MBTL1JAK2JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0901474-A1 ARYL PYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1999-03-17 EP disclosed
WO-1997044326-A1 ARYL PYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1997-11-27 WO disclosed