SCHEMBL8470540

SCHEMBL8470540

Nc1nc2c(cnn2CCC(O)c2ccc(O)c(I)c2)c2nc(-c3ccco3)nn12

nearest known ligand 0.65

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 13/20 0.62
ADORA1 P30542 7/20 0.58
KDM4E B2RXH2 1/20 0.58
NPC1 O15118 1/20 0.58
ALDH1A1 P00352 1/20 0.58
TP53 P04637 1/20 0.58
CYP3A4 P08684 1/20 0.58
ADORA3 P0DMS8 1/20 0.58
HPGD P15428 1/20 0.58
ALOX15 P16050 1/20 0.58
MAPK1 P28482 1/20 0.58
ADORA2B P29275 1/20 0.58
RAB9A P51151 1/20 0.58
SMN1; SMN2 Q16637 1/20 0.58
HSD17B10 Q99714 1/20 0.58
HDAC1 Q13547 1/20 0.55
HDAC6 Q9UBN7 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7344952 0.85 ADORA2A (0.77) ADORA2AADORA1KDM4ENPC1ALDH1A1
SCHEMBL8124748 0.83 ADORA2A (0.85) ADORA2AADORA1HPGD
SCHEMBL7333945 0.80 ADORA2A (0.71) ADORA2AADORA1KDM4ENPC1ALDH1A1
SCHEMBL7346016 0.78 ADORA2A (0.90) ADORA2AADORA1KDM4ENPC1ALDH1A1
SCHEMBL4759580 0.78 ADORA2A (0.76) ADORA2AADORA1KDM4ENPC1ALDH1A1
SCHEMBL12972222 0.77 ADORA2A (0.77) ADORA2AADORA1KDM4ENPC1ALDH1A1
SCHEMBL7343382 0.76 ADORA2A (0.75) ADORA2AADORA1KDM4ENPC1ALDH1A1
SCHEMBL13904673 0.76 ADORA2A (0.76) ADORA2AADORA1KDM4ENPC1ALDH1A1
SCHEMBL13853059 0.76 ADORA2A (0.76) ADORA2AADORA1KDM4ENPC1ALDH1A1
SCHEMBL7339226 0.75 ADORA2A (1.00) ADORA2AADORA1KDM4ENPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5935964-A 1,2,4-triazolo 1,5-c! pyrimidine heterocyclic analogues having antagonistic activity on adenosine A2a receptor SCHERING CORPORATION (US) 1999-08-10 US disclosed