SCHEMBL8477520

SCHEMBL8477520

Cc1cc(C)cc(-c2c([C@H](C)CO)c3cc(C(C)(C)C(=O)N4CC5CCC4CC5)cnc3n2C(=O)OC(C)(C)C)c1

nearest known ligand 0.50

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 1/20 0.50
GNRHR P30968 19/20 0.44
CYP3A4 P08684 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8477523 1.00 CACNA1B (0.50) CACNA1BGNRHRCYP3A4
SCHEMBL8479459 0.94 GNRHR (0.44) CACNA1BGNRHRCYP3A4
SCHEMBL8479454 0.94 GNRHR (0.44) CACNA1BGNRHRCYP3A4
SCHEMBL8183827 0.91 CACNA1B (0.54) CACNA1BGNRHRCYP3A4
SCHEMBL8183825 0.91 CACNA1B (0.54) CACNA1BGNRHRCYP3A4
SCHEMBL8479412 0.88 GNRHR (0.44) GNRHRCYP3A4
SCHEMBL7987363 0.85 CACNA1B (0.52) CACNA1BGNRHRCYP3A4
SCHEMBL7980867 0.84 CACNA1B (0.46) CACNA1BGNRHRCYP3A4
SCHEMBL7980869 0.84 CACNA1B (0.46) CACNA1BGNRHRCYP3A4
SCHEMBL8523626 0.83 GNRHR (0.54) GNRHRCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5998432-A SEXUAL DISORDERS MERCK & CO., INC. (US) 1999-12-07 US disclosed