SCHEMBL8479045

SCHEMBL8479045

O=C1CCCC(CCC2CCCCO2)(c2ccc(Cl)c(Cl)c2)CN1Cc1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.45

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 19/20 0.45
TACR2 P21452 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8487498 0.83 TACR1 (0.51) TACR1TACR2
SCHEMBL8484370 0.82 TACR1 (0.50) TACR1TACR2
SCHEMBL7765734 0.78 TACR1 (0.40) TACR1TACR2
SCHEMBL8485327 0.78 TACR1 (0.46) TACR1TACR2
SCHEMBL8483549 0.77 TACR1 (0.56) TACR1TACR2
SCHEMBL8483945 0.76 TACR1 (0.55) TACR1TACR2
SCHEMBL8991937 0.75 TACR1 (0.48) TACR1TACR2
SCHEMBL22901986 0.74 TACR1 (0.63) TACR1TACR2
SCHEMBL8991959 0.74 TACR1 (0.63) TACR1TACR2
Water SCHEMBL8840361 0.74 TACR1 (0.47) TACR1TACR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5859029-A TREATING SUBSTANCE P-DEPENDENT PATHOLOGICAL CONDITIONS SANOFI (FR) 1999-01-12 US disclosed
US-5656639-A POSSESS STRONG AFFINITY FOR NK1 RECEPTORS; USEFUL IN TREATMENT OF SUBSTANCE P-DEPENDENT PATHOLOGICAL CONDITIONS SANOFI (FR) 1997-08-12 US disclosed
EP-0723959-A1 Heterocyclic compounds as tachykinin receptor antagonists, process for their preparation and pharmaceuticals containing them SANOFI (FR) 1996-07-31 EP disclosed