SCHEMBL8482175

SCHEMBL8482175

O=C(c1cc(C(F)(F)F)cc(C(F)(F)F)c1)N1CCN(CCCCCc2ccccc2)C[C@H]1Cc1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 15/20 0.58
CA1 P00915 2/20 0.48
CA2 P00918 2/20 0.48
CA4 P22748 2/20 0.48
CA9 Q16790 2/20 0.48
SIGMAR1 Q99720 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8475591 0.99 TACR1 (0.57) TACR1CA1CA2CA4CA9
Hydrochloric Acid SCHEMBL8475949 0.98 TACR1 (0.58) TACR1CA1CA2CA4CA9
SCHEMBL9238709 0.88 TACR1 (0.55) TACR1CA1CA2CA4CA9
Hydrochloric Acid SCHEMBL8481763 0.87 TACR1 (0.55) TACR1CA1CA2CA4CA9
Hydrochloric Acid SCHEMBL8480341 0.87 TACR1 (0.50) TACR1CA1CA2CA4CA9
Hydrochloric Acid SCHEMBL9241462 0.87 TACR1 (0.50) TACR1CA1CA2CA4CA9
Hydrochloric Acid SCHEMBL8480614 0.86 TACR1 (0.55) TACR1CA1CA2CA4CA9
SCHEMBL8481079 0.86 TACR1 (0.64) TACR1CA1CA2CA4CA9
Hydrochloric Acid SCHEMBL8479202 0.85 TACR1 (0.63) TACR1CA1CA2CA4CA9
Hydrochloric Acid SCHEMBL8480502 0.85 TACR1 (0.58) TACR1CA1CA2CA4CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5883098-A USED AS TACHYKININ ANTAGONISTS IN THE TREATMENT OF RESPIRATORY DISEASES, OPHTHALMIC DISEASES AND INFLAMMATORY DISEASES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1999-03-16 US disclosed
US-5670505-A TACHYKIKIN ANTAGONIST FOR RESPIRATORY DISEASES, OPHTHALMIC DISEASES AND ANTIINFLAMMATORY AGENTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-09-23 US disclosed
EP-0655442-A1 Piperazine derivatives as Tachykinin antagonists FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1995-05-31 EP disclosed