SCHEMBL8484386

SCHEMBL8484386

COc1cccc(CNCC(CCN2CCC(NC(C)=O)(c3ccccc3)CC2)c2ccc(Cl)c(Cl)c2)c1

nearest known ligand 0.60

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TACR2 P21452 6/20 0.60
TACR1 P25103 4/20 0.60
TACR3 P29371 7/20 0.55
MCHR1 Q99705 1/20 0.48
CCR5 P51681 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8482751 0.87 TACR2 (0.67) TACR2TACR1TACR3CCR5
SCHEMBL8482847 0.85 TACR2 (0.66) TACR2TACR1TACR3CCR5
SCHEMBL6950402 0.84 TACR1 (0.61) TACR2TACR1TACR3
SCHEMBL7870009 0.82 TACR2 (0.73) TACR2TACR1TACR3
SCHEMBL14089179 0.81 TACR2 (0.75) TACR2TACR1TACR3
SCHEMBL6952599 0.80 TACR2 (0.73) TACR2TACR1TACR3
SCHEMBL7864418 0.80 TACR2 (0.65) TACR2TACR1TACR3CCR5
SCHEMBL7312636 0.79 TACR2 (0.66) TACR2TACR1TACR3
Hydrochloric Acid SCHEMBL7751882 0.78 TACR2 (0.65) TACR2TACR1TACR3
SCHEMBL8478954 0.78 TACR2 (0.72) TACR2TACR1TACR3CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6008223-A ANTIINFLAMMATORY AGENTS FOR TREATING ASTHMA ZENECA LIMITED (GB) 1999-12-28 US disclosed
US-5731309-A Substituted heteroalkyleneamine neurokinin antagonists ZENECA LIMITED (GB) 1998-03-24 US disclosed