SCHEMBL8486941

SCHEMBL8486941

CN(C)CCn1nc2c3c(c(N)ccc31)Sc1ncccc1-2

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 14/20 0.36
TOP2B Q02880 2/20 0.33
NQO1 P15559 1/20 0.32
GSK3B P49841 1/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
KDM4E B2RXH2 1/20 0.31
FYN P06241 1/20 0.31
YES1 P07947 1/20 0.31
LYN P07948 1/20 0.31
FGR P09769 1/20 0.31
SRC P12931 1/20 0.31
KDM1A O60341 1/20 0.30
NPC1 O15118 1/20 0.30
MITF O75030 1/20 0.30
POLB P06746 1/20 0.30
DNMT1 P26358 1/20 0.30
HTT P42858 1/20 0.30
RAD52 P43351 1/20 0.30
RAB9A P51151 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8486027 0.86 TOP2A (0.32) TOP2A
SCHEMBL8486726 0.85 TOP2A (0.32) TOP2ATOP2B
SCHEMBL8483875 0.84 KDM1A (0.34) TOP2ATOP2BGSK3BSMN1; SMN2KDM4E
SCHEMBL10925471 0.84 TOP2A (0.39) TOP2ATOP2BSMN1; SMN2KDM4EKDM1A
SCHEMBL8485663 0.80 TOP2A (0.46) TOP2A
SCHEMBL8721611 0.79 TOP2A (0.49) TOP2ATOP2B
SCHEMBL8485118 0.79 CYP2D6 (0.36) TOP2ATOP2BNQO1GSK3B
SCHEMBL8483006 0.79 TOP2A (0.37) TOP2ATOP2BNQO1GSK3B
SCHEMBL8721606 0.79 TOP2A (0.35) TOP2ATOP2B
SCHEMBL10812739 0.78 CYP1A2 (0.40) TOP2ATOP2BNQO1GSK3BSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5935969-A Pyrido-thiopyrandoinazoles with antitumor activity UNIVERSITY OF VERMONT (US) 1999-08-10 US disclosed