SCHEMBL8488117

SCHEMBL8488117

COC(=O)Cc1c[nH]cc1CC(=O)OC

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AB1 P08238 1/20 0.47
CYP4F2 P78329 1/20 0.44
CYP4A11 Q02928 1/20 0.44
ALDH1A1 P00352 5/20 0.42
KDM4E B2RXH2 4/20 0.42
HSD17B10 Q99714 3/20 0.42
MAPT P10636 3/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
TSHR P16473 3/20 0.42
TP53 P04637 1/20 0.41
GAA P10253 3/20 0.39
EGFR P00533 1/20 0.39
GLA P06280 1/20 0.39
PDGFRB P09619 1/20 0.39
FGFR1 P11362 1/20 0.39
PDGFRA P16234 1/20 0.39
FLT1 P17948 1/20 0.39
FGFR3 P22607 1/20 0.39
KDR P35968 1/20 0.39
GFER P55789 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8151890 0.87 HSP90AB1 (0.46) HSP90AB1CYP4F2CYP4A11ALDH1A1KDM4E
SCHEMBL27451821 0.86 HSP90AB1 (0.44) HSP90AB1CYP4F2CYP4A11ALDH1A1KDM4E
SCHEMBL970536 0.84 PDGFRB (0.47) HSP90AB1CYP4F2CYP4A11ALDH1A1KDM4E
SCHEMBL14354674 0.80 HSP90AB1 (0.56) HSP90AB1CYP4F2CYP4A11ALDH1A1KDM4E
SCHEMBL970569 0.78 KMT2A (0.45) ALDH1A1KDM4EHSD17B10MAPTSMN1; SMN2
SCHEMBL14565681 0.77 HSP90AB1 (0.44) HSP90AB1CYP4F2CYP4A11ALDH1A1KDM4E
SCHEMBL1554320 0.76 KDM4E (0.53) HSP90AB1CYP4F2CYP4A11ALDH1A1KDM4E
SCHEMBL13283682 0.74 HSP90AB1 (0.55) HSP90AB1CYP4F2CYP4A11ALDH1A1KDM4E
SCHEMBL951010 0.73 PDGFRB (0.41) HSP90AB1CYP4F2CYP4A11ALDH1A1KDM4E
SCHEMBL104485 0.73 KMT2A (0.51) MAPTSMN1; SMN2GAALMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5877165-A CONTAINING MULTIPLE CARBORANE CAGES WHICH SELECTIVELY ACCUMULATE IN NEOPLASTIC TISSUE WITHIN THE IRRADIATION VOLUME AND THUS CAN BE USED IN CANCER THERAPIES SUCH AS BORON NEUTRON CAPTURE THERAPY AND PHOTODYNAMIC THERAPY. BROOKHAVEN SCIENCE ASSOCIATES (US) 1999-03-02 US disclosed