SCHEMBL8501030

SCHEMBL8501030

CC(C(=O)O)c1ccc(Oc2c(-c3cccc(O)c3)ccc3cc(O)ccc23)cc1

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 8/20 0.54
AKR1C2 P52895 8/20 0.54
ESR1 P03372 8/20 0.53
ESR2 Q92731 8/20 0.53
PTGS2 P35354 4/20 0.41
AKR1C4 P17516 1/20 0.41
AKR1C1 Q04828 1/20 0.41
PTGS1 P23219 3/20 0.41
CDC42 P60953 1/20 0.41
RAC1 P63000 1/20 0.41
CYP1A2 P05177 1/20 0.41
TSHR P16473 1/20 0.41
SLC22A6 Q4U2R8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8497703 0.93 AKR1C3 (0.52) AKR1C3AKR1C2ESR1ESR2PTGS2
SCHEMBL8498073 0.92 ESR1 (0.57) AKR1C3AKR1C2ESR1ESR2PTGS2
SCHEMBL8500571 0.92 AKR1C3 (0.55) AKR1C3AKR1C2ESR1ESR2PTGS2
SCHEMBL8499726 0.92 AKR1C3 (0.54) AKR1C3AKR1C2ESR1ESR2PTGS2
SCHEMBL8499781 0.90 ESR1 (0.51) AKR1C3AKR1C2ESR1ESR2PTGS2
SCHEMBL8497551 0.87 APP (0.54) AKR1C3AKR1C2ESR1ESR2PTGS2
SCHEMBL8502302 0.87 ESR1 (0.53) AKR1C3AKR1C2ESR1ESR2AKR1C1
SCHEMBL8497872 0.86 ESR1 (0.54) AKR1C3AKR1C2ESR1ESR2PTGS2
SCHEMBL8500226 0.86 ESR1 (0.46) AKR1C3AKR1C2ESR1ESR2PTGS2
SCHEMBL8500476 0.86 ESR1 (0.48) AKR1C3AKR1C2ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5916916-A USEFUL AS SELECTIVE ESTROGEN RECEPTOR MODULATORS. ELI LILLY AND COMPANY (US) 1999-06-29 US claimed
US-5916916-A USEFUL AS SELECTIVE ESTROGEN RECEPTOR MODULATORS. ELI LILLY AND COMPANY (US) 1999-06-29 US disclosed