SCHEMBL8501417

SCHEMBL8501417

COc1ccc2c(Oc3ccc(C(C)C(=O)O)cc3)c(-c3ccc(OC)c(F)c3)ccc2c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APP P05067 2/20 0.52
CYP2C19 P33261 1/20 0.52
AKR1C3 P42330 14/20 0.50
AKR1C2 P52895 14/20 0.50
PTGS2 P35354 4/20 0.50
PTGS1 P23219 2/20 0.50
CDC42 P60953 1/20 0.50
RAC1 P63000 1/20 0.50
CYP1A2 P05177 1/20 0.50
TSHR P16473 1/20 0.50
SLC22A6 Q4U2R8 1/20 0.50
AKR1C4 P17516 1/20 0.42
AKR1C1 Q04828 1/20 0.42
PSEN1 P49768 1/20 0.40
PSEN2 P49810 1/20 0.40
APH1B Q8WW43 1/20 0.40
NCSTN Q92542 1/20 0.40
APH1A Q96BI3 1/20 0.40
PSENEN Q9NZ42 1/20 0.40
FFAR1 O14842 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8501435 0.88 APP (0.56) APPCYP2C19AKR1C3AKR1C2PTGS2
SCHEMBL8497582 0.88 AKR1C3 (0.59) APPCYP2C19AKR1C3AKR1C2PTGS2
SCHEMBL8497441 0.85 AKR1C3 (0.55) APPCYP2C19AKR1C3AKR1C2PTGS2
SCHEMBL8501466 0.85 AKR1C3 (0.55) APPCYP2C19AKR1C3AKR1C2PTGS2
SCHEMBL8502209 0.85 AKR1C3 (0.59) APPCYP2C19AKR1C3AKR1C2PTGS2
SCHEMBL8501245 0.84 AKR1C3 (0.54) APPCYP2C19AKR1C3AKR1C2PTGS2
SCHEMBL8498571 0.83 AKR1C3 (0.40) AKR1C3AKR1C2FFAR1
SCHEMBL7200140 0.83 ESR1 (0.49)
SCHEMBL7200144 0.83 ESR1 (0.49)
SCHEMBL8497703 0.82 AKR1C3 (0.52) APPCYP2C19AKR1C3AKR1C2PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5916916-A USEFUL AS SELECTIVE ESTROGEN RECEPTOR MODULATORS. ELI LILLY AND COMPANY (US) 1999-06-29 US claimed
US-5916916-A USEFUL AS SELECTIVE ESTROGEN RECEPTOR MODULATORS. ELI LILLY AND COMPANY (US) 1999-06-29 US disclosed