SCHEMBL8517279

SCHEMBL8517279

CC/C=C/[C@H]1CC[C@H](CCc2cnc(-c3ccc(F)c(Cl)c3)nc2)CC1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 2/20 0.34
TGFBR1 P36897 4/20 0.33
TGFBR2 P37173 3/20 0.33
CHRNB1 P11230 1/20 0.33
CHRNB2 P17787 1/20 0.33
CHRNB4 P30926 1/20 0.33
CHRNA3 P32297 1/20 0.33
CHRNB3 Q05901 1/20 0.33
RXRA P19793 1/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2B Q13224 1/20 0.32
ACACB O00763 1/20 0.31
CNR1 P21554 1/20 0.31
CYP11B1 P15538 1/20 0.31
CYP11B2 P19099 1/20 0.31
CHRM3 P20309 3/20 0.31
AXL P30530 1/20 0.31
SLC5A2 P31639 1/20 0.31
CHRM2 P08172 1/20 0.30
CHRM1 P11229 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9313047 1.00 GRM2 (0.34) GRM2TGFBR1TGFBR2CHRNB1CHRNB2
SCHEMBL8517283 1.00 GRM2 (0.34) GRM2TGFBR1TGFBR2CHRNB1CHRNB2
SCHEMBL9312823 0.92 GRM2 (0.33) GRM2TGFBR1TGFBR2CHRNB1CHRNB2
SCHEMBL9312833 0.92 GRM2 (0.33) GRM2TGFBR1TGFBR2CHRNB1CHRNB2
SCHEMBL9312838 0.92 GRM2 (0.33) GRM2TGFBR1TGFBR2CHRNB1CHRNB2
SCHEMBL9312835 0.92 GRM2 (0.33) GRM2TGFBR1TGFBR2CHRNB1CHRNB2
SCHEMBL9311776 0.92 SLC5A2 (0.33) ACACBCYP11B1CYP11B2SLC5A2
SCHEMBL9311767 0.92 SLC5A2 (0.33) ACACBCYP11B1CYP11B2SLC5A2
SCHEMBL9311781 0.92 SLC5A2 (0.33) ACACBCYP11B1CYP11B2SLC5A2
SCHEMBL8517354 0.91 PDGFRB (0.31) SLC5A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0475273-B1 Liquid crystal mixture containing halogenated alcenyl compounds MERCK PATENT GMBH (DE) 1999-04-07 EP disclosed
US-5292452-A Electrooptical devices; high dielectric anisotropy, low rotation viscosity, short response time HOFFMANN-LA ROCHE INC. (US) 1994-03-08 US disclosed
EP-0475273-A1 Halogenated alcenyl compounds F. HOFFMANN-LA ROCHE AG (CH) 1992-03-18 EP disclosed