Ethyne

Ethyne

SCHEMBL8517660

C#C.OCC1CCCC1O

nearest known ligand 0.44

Full drug profile on Sugi Atlas →

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA4 P22748 1/20 0.44
TDP1 Q9NUW8 1/20 0.35
GBA1 P04062 5/20 0.34
PYGL P06737 1/20 0.34
GBA2 Q9HCG7 1/20 0.34
GAA P10253 1/20 0.34
GLB1 P16278 1/20 0.34
PTGS1 P23219 7/20 0.33
PTGS2 P35354 6/20 0.33
MT-CO1 P00395 1/20 0.33
MT-CO2 P00403 1/20 0.33
PABPC1 P11940 1/20 0.32
APOBEC3A P31941 1/20 0.32
APOBEC3G Q9HC16 1/20 0.32
AGL P35573 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL260593 0.95
SCHEMBL7091680 0.95
SCHEMBL26008596 0.95
SCHEMBL7091682 0.95
SCHEMBL10433294 0.95
SCHEMBL24814038 0.95
SCHEMBL27786042 0.92
Ethane SCHEMBL27566965 0.90 CA1 (0.50) CA1CA2CA4TDP1GBA1
SCHEMBL898707 0.89
SCHEMBL18462018 0.89

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5977325-A NUCLEOSIDE DERIVATIVES USEFUL AS ANTICARCINOGENIC/ANTITUMOR AGENTS AND VIRICIDES MERRELL PHARMACEUTICALS INC. (US) 1999-11-02 US disclosed
US-5616702-A ANTITUMOR AGENTS, VIRICIDES MERRELL PHARMACEUTICALS INC. (US) 1997-04-01 US disclosed
US-5607925-A Treatment of carcinoma by administration of 2'-halomethylidenyl-2'-deoxynucleosides MERRELL PHARMACEUTICALS INC. (US) 1997-03-04 US disclosed
US-5378693-A Antitumor agents or viricides MERRELL DOW PHARMACEUTICALS INC. (US) 1995-01-03 US disclosed
EP-0372268-B1 Novel 2'-halomethylidene, 2'-ethenylidene and 2'-ethynyl cytidine, uridine and guanosine derivatives MERRELL DOW PHARMA (US) 1994-05-04 EP disclosed
EP-0372268-A1 Novel 2'-halomethylidene, 2'-ethenylidene and 2'-ethynyl cytidine, uridine and guanosine derivatives MERRELL DOW PHARMACEUTICALS INC. (US) 1990-06-13 EP disclosed