SCHEMBL8519542

SCHEMBL8519542

COC(=O)c1ccc(NC(=O)C(O)c2ccc3c(c2)C(C)(C)CCC3(C)C)c(F)c1

nearest known ligand 0.81

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARB P10826 10/20 0.81
RARG P13631 10/20 0.81
CYP3A4 P08684 7/20 0.81
CYP26A1 O43174 6/20 0.81
RXRA P19793 3/20 0.46
RXRB P28702 2/20 0.44
RARA P10276 9/20 0.43
CYP26B1 Q9NR63 1/20 0.43
NPC1 O15118 1/20 0.42
LMNA P02545 1/20 0.42
MAPT P10636 1/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
ALDH1A1 P00352 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
TSHR P16473 1/20 0.38
MAPK1 P28482 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29354207 0.89 RARB (1.00) RARBRARGCYP3A4CYP26A1RXRA
SCHEMBL29613246 0.89 RARB (1.00) RARBRARGCYP3A4CYP26A1RXRA
SCHEMBL30477013 0.89 RARB (1.00) RARBRARGCYP3A4CYP26A1RXRA
SCHEMBL3756112 0.89 RARB (1.00) RARBRARGCYP3A4CYP26A1RXRA
SCHEMBL165751 0.89 RARB (1.00) RARBRARGCYP3A4CYP26A1RXRA
SCHEMBL165750 0.89 RARB (1.00) RARBRARGCYP3A4CYP26A1RXRA
SCHEMBL2788640 0.75 CYP3A4 (0.70) RARBRARGCYP3A4CYP26A1RXRA
SCHEMBL5080286 0.74 RARB (0.71) RARBRARGCYP3A4CYP26A1RXRA
SCHEMBL8839311 0.74 RARG (0.50) RARBRARGCYP3A4CYP26A1RXRA
SCHEMBL6343446 0.71 CYP3A4 (0.44) RARBRARGCYP3A4CYP26A1RXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0747347-B1 RAR-gamma-specific retinobenzoic acid derivatives BRISTOL MYERS SQUIBB CO (US) 1999-07-21 EP disclosed
US-5624957-A RETINOID ACTIVE COMPOUNDS BRISTOL-MYERS SQUIBB COMPANY (US) 1997-04-29 US disclosed
EP-0747347-A1 RARy-specific retinobenzoic acid derivatives BRISTOL-MYERS SQUIBB COMPANY (US) 1996-12-11 EP disclosed