SCHEMBL8520119

SCHEMBL8520119

COC(=O)Oc1ccc2cncnc2c1

nearest known ligand 0.65

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
EGFR P00533 5/20 0.65
IMPDH2 P12268 1/20 0.46
HPGDS O60760 12/20 0.45
NOTUM Q6P988 1/20 0.44
BAZ1A Q9NRL2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27630991 0.85 EGFR (0.64) EGFRIMPDH2HPGDSNOTUM
SCHEMBL7513856 0.83 EGFR (0.61) EGFRIMPDH2HPGDSNOTUMBAZ1A
SCHEMBL6825418 0.82 EGFR (0.59) EGFRIMPDH2HPGDSNOTUMBAZ1A
SCHEMBL29517021 0.79 EGFR (1.00) EGFRHPGDS
SCHEMBL30241125 0.79 EGFR (1.00) EGFRHPGDS
SCHEMBL668493 0.79 EGFR (1.00) EGFRHPGDS
Hydrochloric Acid SCHEMBL28023744 0.78 EGFR (0.96) EGFRHPGDS
SCHEMBL8414749 0.77 CYP3A4 (0.51) IMPDH2
SCHEMBL2944091 0.77 KDM4E (0.47)
SCHEMBL30507829 0.76 CSNK2A1 (0.59) EGFRIMPDH2NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0927192-A1 MODIFIED AMINOACIDS, PHARMACEUTICALS CONTAINING THESE COMPOUNDS AND METHOD FOR THEIR PRODUCTION Dr. Karl Thomae GmbH (DE) 1999-07-07 EP disclosed
WO-1998011128-A1 MODIFIED AMINOACIDS, PHARMACEUTICALS CONTAINING THESE COMPOUNDS AND METHOD FOR THEIR PRODUCTION DR. KARL THOMAE GMBH (DE) 1998-03-19 WO disclosed