SCHEMBL8522666

SCHEMBL8522666

COc1c(OCCOC2CCCCO2)cccc1ON(c1ccccc1)S(=O)(=O)c1ccc(C(C)(C)C)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.35
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
NPSR1 Q6W5P4 1/20 0.35
GAA P10253 2/20 0.34
MAPT P10636 1/20 0.34
EDNRA P25101 5/20 0.33
PSEN1 P49768 2/20 0.33
PSEN2 P49810 2/20 0.33
APH1B Q8WW43 2/20 0.33
NCSTN Q92542 2/20 0.33
APH1A Q96BI3 2/20 0.33
PSENEN Q9NZ42 2/20 0.33
SPPL2A Q8TCT8 1/20 0.33
EDNRB P24530 3/20 0.33
USP2 O75604 1/20 0.33
HTR1A P08908 1/20 0.33
DRD2 P14416 1/20 0.33
HTR2A P28223 1/20 0.33
HTR7 P34969 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7568861 0.76 EDNRA (0.52) EDNRAEDNRB
SCHEMBL8522671 0.76 ITGB1 (0.35) EDNRAEDNRBKDM4CNPC1RAB9A
SCHEMBL7568989 0.69 EDNRA (0.56) EDNRAEDNRB
SCHEMBL7567982 0.68 NPC1 (0.44) ALDH1A1MEN1KMT2AMAPTHTR1A
SCHEMBL7814508 0.67 EDNRA (0.59) EDNRAEDNRB
SCHEMBL7566546 0.67 KDM4C (0.40) ALDH1A1MEN1KMT2AHTR1AKDM4C
SCHEMBL11168223 0.66 MEN1 (0.44) ALDH1A1MEN1KMT2AMAPTKDM4C
SCHEMBL12510434 0.65 MEN1 (0.49) ALDH1A1MEN1KMT2AMAPTKDM4C
SCHEMBL871773 0.65 KMT2A (0.55) ALDH1A1MEN1KMT2AKDM4C
SCHEMBL8354599 0.65 KDM4C (0.38) MEN1KMT2AKDM4CNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5962682-A Aryl- and hetaryl-sulfonamide derivatives, their preparation and their use as endothelin antagonists HOFFMANN-LA ROCHE INC. (US) 1999-10-05 US disclosed