SCHEMBL8527002

SCHEMBL8527002

N[C@H](Cc1ccccc1)CS(=O)(=O)O

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.59
ANPEP P15144 2/20 0.52
ALPI P09923 1/20 0.50
PKM P14618 1/20 0.50
PTGS1 P23219 1/20 0.50
XIAP P98170 1/20 0.50
SLC7A5 Q01650 1/20 0.50
MMP2 P08253 3/20 0.47
LAP3 P28838 3/20 0.47
SLC1A3 P43003 1/20 0.46
SLC1A2 P43004 1/20 0.46
SLC1A1 P43005 1/20 0.46
SLC6A2 P23975 2/20 0.45
TAAR1 Q96RJ0 2/20 0.45
MAOA P21397 1/20 0.45
SLC6A4 P31645 1/20 0.45
SLC6A3 Q01959 1/20 0.45
SIGMAR1 Q99720 1/20 0.45
CYP2A6 P11509 1/20 0.45
ADORA2A P29274 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27712365 1.00 EPHX1 (0.59) EPHX1ANPEPALPIPKMPTGS1
SCHEMBL6033692 1.00 EPHX1 (0.59) EPHX1ANPEPALPIPKMPTGS1
Hydrochloric Acid SCHEMBL29410716 0.98 EPHX1 (0.57) EPHX1ANPEPALPIPKMPTGS1
SCHEMBL8748122 0.83 TAAR1 (0.50) SLC7A5SLC6A2TAAR1
SCHEMBL18167808 0.82 EPHX1 (0.61) EPHX1ANPEPALPIPKMPTGS1
SCHEMBL18167806 0.82 EPHX1 (0.61) EPHX1ANPEPALPIPKMPTGS1
SCHEMBL27700316 0.81 ANPEP (0.50) EPHX1ANPEP
SCHEMBL27720875 0.81 EPHX1 (0.55) EPHX1ANPEPALPIPKMPTGS1
SCHEMBL352772 0.81 EPHX1 (0.55) EPHX1ANPEPALPIPKMPTGS1
SCHEMBL27700318 0.81 EPHX1 (0.55) EPHX1ANPEPALPIPKMPTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101103969-A Therapeutic formulations for the treatment of beta-amyloid related diseases NEUROCHEM INTERNAT LTD (CH) 2008-01-16 CN disclosed
EP-0460679-B1 Endothelin antagonistic peptide derivatives BANYU PHARMA CO LTD (JP) 1998-10-28 EP disclosed
US-5691315-A CARDIOVASCULAR DISORDERS; VASODILATOR; BRONCHODILATOR BANYU PHARMACEUTICAL CO., LTD. (JP) 1997-11-25 US disclosed
US-5470833-A Vasodilators, bronchodilators BANYU PHARMACEUTICAL CO., LTD. (JP) 1995-11-28 US disclosed
US-5444152-A Vasolidator or bronchodilator BANYU PHARMACEUTICAL CO., LTD. (JP) 1995-08-22 US disclosed
EP-0460679-A2 Endothelin antagonistic peptide derivatives Banyu Pharmaceutical Co., Ltd. (JP) 1991-12-11 EP disclosed