SCHEMBL8529147

SCHEMBL8529147

CC(C)(C)C(=Cc1ccccc1)C(N)=O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 1/20 0.49
TSHR P16473 2/20 0.47
NPC1 O15118 1/20 0.47
AKR1C3 P42330 1/20 0.47
CYP2C19 P33261 1/20 0.44
KMT2A Q03164 2/20 0.42
ALDH1A1 P00352 2/20 0.42
MAPT P10636 2/20 0.42
AKR1C1 Q04828 1/20 0.41
RECQL P46063 1/20 0.41
MEN1 O00255 1/20 0.41
HTT P42858 1/20 0.40
EGFR P00533 1/20 0.40
FBP1 P09467 2/20 0.39
KDM4E B2RXH2 1/20 0.39
LMNA P02545 1/20 0.39
HPGD P15428 1/20 0.39
GLA P06280 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
CYP3A4 P08684 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL525211 0.84 AKR1C3 (0.55) TSHRNPC1AKR1C3CYP2C19KMT2A
SCHEMBL525210 0.84 AKR1C3 (0.55) TSHRNPC1AKR1C3CYP2C19KMT2A
SCHEMBL28499934 0.83 GRIN2D (0.42) NPC1AKR1C3KMT2AALDH1A1MAPT
SCHEMBL10625434 0.82 AKR1C3 (0.53) TSHRNPC1AKR1C3CYP2C19KMT2A
SCHEMBL28501761 0.81 CYP2C9 (0.51) AKR1C3ALDH1A1AKR1C1HTTFBP1
SCHEMBL6510379 0.81 MCL1 (0.49) MCL1TSHRNPC1AKR1C3CYP2C19
SCHEMBL7564827 0.81 MCL1 (0.49) MCL1TSHRNPC1AKR1C3CYP2C19
SCHEMBL1291048 0.79 MCL1 (0.47) MCL1TSHRAKR1C3KMT2AALDH1A1
SCHEMBL13108767 0.77 EGFR (0.51) TSHRNPC1AKR1C3CYP2C19KMT2A
SCHEMBL13123943 0.77 EGFR (0.51) TSHRNPC1AKR1C3CYP2C19KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998042657-A1 SYNTHESIS OF α,β-SUBSTITUTED AMINO AMIDES, ESTERS AND ACIDS THE SCRIPPS RESEARCH INSTITUTE (US) 1998-10-01 WO disclosed