SCHEMBL8530402

SCHEMBL8530402

CC(NC(=O)OCc1ccccc1)c1ccccc1

nearest known ligand 0.68

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ATM Q13315 2/20 0.68
CYP3A4 P08684 6/20 0.65
TSHR P16473 6/20 0.65
CTSL P07711 1/20 0.59
CTSS P25774 1/20 0.59
CTSK P43235 2/20 0.57
MMP9 P14780 1/20 0.56
CTRB1 P17538 2/20 0.56
ALDH1A1 P00352 3/20 0.56
CYP1A2 P05177 2/20 0.56
ELANE P08246 1/20 0.56
CYP2C9 P11712 4/20 0.55
CYP2C19 P33261 3/20 0.55
POLB P06746 1/20 0.55
CYP2D6 P10635 1/20 0.55
LMNA P02545 1/20 0.55
MEN1 O00255 1/20 0.55
KMT2A Q03164 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21469067 1.00 ATM (0.68) ATMCYP3A4TSHRCTSLCTSS
SCHEMBL30460502 1.00 ATM (0.68) ATMCYP3A4TSHRCTSLCTSS
SCHEMBL13721922 0.92 ATM (0.63) ATMCYP3A4TSHRCTSLCTSS
SCHEMBL18459501 0.92 ATM (0.63) ATMCYP3A4TSHRCTSLCTSS
SCHEMBL13721804 0.92 ATM (0.63) ATMCYP3A4TSHRCTSLCTSS
SCHEMBL4444864 0.90 ATM (0.60) ATMCYP3A4TSHRCTSLCTSS
SCHEMBL21399863 0.90 ATM (0.60) ATMCYP3A4TSHRCTSLCTSS
SCHEMBL2851560 0.90 ATM (0.60) ATMCYP3A4TSHRCTSLCTSS
SCHEMBL12951666 0.90 ATM (0.60) ATMCYP3A4TSHRCTSLCTSS
SCHEMBL21404926 0.90 ATM (0.60) ATMCYP3A4TSHRCTSLCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3013812-B1 KAPPA OPIOID AGONISTS AND USES THEREOF NEKTAR THERAPEUTICS (US) 2019-10-16 EP disclosed
US-7449447-B2 Peptidomimetic NS3-serine protease inhibitors of hepatitis C virus SCHERING CORPORATION (US) 2008-11-11 US disclosed
US-5807875-A OBESITY THERAPY DR. KARL THOMAE GMBH (DE) 1998-09-15 US disclosed