SCHEMBL8530877

SCHEMBL8530877

O=C(Nc1ccc(F)c(C(F)(F)F)c1)C(F)(F)F

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 3/20 0.58
GRM4 Q14833 1/20 0.57
CYP1A2 P05177 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.50
KDR P35968 1/20 0.50
CDK8 P49336 1/20 0.48
BLM P54132 1/20 0.48
WRN Q14191 1/20 0.48
GAA P10253 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
KCNQ3 O43525 1/20 0.47
KCNQ2 O43526 1/20 0.47
KCNE1 P15382 1/20 0.47
KCNQ1 P51787 1/20 0.47
PGR P06401 1/20 0.47
CYP3A4 P08684 1/20 0.47
SLC22A12 Q96S37 1/20 0.47
CA12 O43570 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9891509 0.87 AR (0.63) ARGRM4L3MBTL1KDRCDK8
SCHEMBL8902443 0.86 CYP1A2 (0.54) ARCYP1A2CYP2C9CYP2C19L3MBTL1
SCHEMBL4123404 0.85 AR (0.64) ARGRM4KDRGAAPGR
SCHEMBL1904289 0.84 AR (0.64) ARGRM4KDRCDK8BLM
SCHEMBL8029788 0.84 AR (0.60) ARGRM4KDRCDK8BLM
SCHEMBL6602968 0.84 CYP1A2 (0.56) CYP1A2CYP2C9CYP2C19L3MBTL1GAA
SCHEMBL31146306 0.84 CYP1A2 (0.56) CYP1A2CYP2C9CYP2C19L3MBTL1GAA
SCHEMBL463590 0.83 AR (0.62) ARGRM4L3MBTL1KDRCDK8
SCHEMBL20560568 0.83 GRM4 (0.61) ARGRM4KDRCDK8BLM
SCHEMBL1380778 0.83 AR (0.58) ARGRM4KDRCDK8BLM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0596358-B1 0-Phenylenediamines containing fluoroakyl(ene) groups and their use as intermediates in the preparation of benzimidazoles BAYER AG (DE) 1998-10-28 EP disclosed
US-5484953-A CHEMICAL INTERMEDIATES FOR BENZIMIDAZOLES FOR INSECTICIDES OR NEMATOCIDES BAYER AKTIENGESELLSCHAFT (DE) 1996-01-16 US disclosed
EP-0596358-A1 0-Phenylenediamines containing fluoroakyl(ene) groups and their use as intermediates in the preparation of benzimidazoles BAYER AG (DE) 1994-05-11 EP disclosed