SCHEMBL8536581

SCHEMBL8536581

COc1ccc(NC(=O)c2ccc(-c3ccc(-c4noc(C)n4)cc3C)cc2)cc1C1CC2CCC(C1)N2C

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 15/20 0.67
HTR1B P28222 10/20 0.67
HTR2A P28223 8/20 0.67
SLC6A4 P31645 4/20 0.67
MEN1 O00255 3/20 0.67
MAPT P10636 3/20 0.67
KMT2A Q03164 3/20 0.67
TDP1 Q9NUW8 3/20 0.67
TP53 P04637 2/20 0.67
CYP3A4 P08684 2/20 0.67
CYP2D6 P10635 2/20 0.67
MAPK1 P28482 2/20 0.67
HSD17B10 Q99714 2/20 0.67
HTR2C P28335 2/20 0.67
HTR1A P08908 2/20 0.67
HTR3E A5X5Y0 1/20 0.67
HTR3B O95264 1/20 0.67
CYP2C9 P11712 1/20 0.67
TSHR P16473 1/20 0.67
NFKB1 P19838 1/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7161726 0.90 HTR1D (0.75) HTR1DHTR1BHTR2ASLC6A4MEN1
SCHEMBL8588295 0.89 HTR1D (0.62) HTR1DHTR1BHTR2ASLC6A4MEN1
SCHEMBL8588239 0.89 HTR1D (0.61) HTR1DHTR1BHTR2ASLC6A4MEN1
SCHEMBL6925638 0.88 HTR1D (0.70) HTR1DHTR1BHTR2ASLC6A4MEN1
Oxalic Acid SCHEMBL6926422 0.88 HTR1D (0.72) HTR1DHTR1BHTR2ASLC6A4MEN1
SCHEMBL8586374 0.87 HTR1D (0.64) HTR1DHTR1BHTR2ASLC6A4MEN1
SCHEMBL8934383 0.87 HTR1D (0.71) HTR1DHTR1BHTR2ASLC6A4MEN1
SCHEMBL8934400 0.85 HTR1D (0.57) HTR1DHTR1BHTR2ASLC6A4MEN1
SCHEMBL8532655 0.84 HTR1D (0.57) HTR1DHTR1BHTR2ASLC6A4MEN1
SCHEMBL8794930 0.82 HTR1D (0.70) HTR1DHTR1BHTR2ASLC6A4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0819126-A1 BIPHENYLAMIDE DERIVATIVES AS 5HT 1D? ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1998-01-21 EP claimed
EP-0819126-A1 BIPHENYLAMIDE DERIVATIVES AS 5HT 1D? ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1998-01-21 EP disclosed
WO-1996031508-A1 BIPHENYLAMIDE DERIVATIVES AS 5HT1D ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1996-10-10 WO disclosed