SCHEMBL8537152

SCHEMBL8537152

CN(c1cc(Cl)ncn1)n1cccc1

nearest known ligand 0.41

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 1/20 0.41
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.33
FGFR4 P22455 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8538197 0.76 SLC6A2 (0.61) SLC6A2NPC1
SCHEMBL937306 0.74 NPC1 (0.44) SLC6A2NPC1FGFR4
SCHEMBL9685872 0.71 NPC1 (0.39) SLC6A2NPC1FGFR4
SCHEMBL8537904 0.69 SLC6A2 (0.40) SLC6A2
SCHEMBL5883439 0.68 POLB (0.46) SLC6A2NPC1
SCHEMBL414257 0.68 CSF1R (0.48) SLC6A2NPC1
SCHEMBL16665315 0.67 FGFR4 (0.37) SLC6A2NPC1FGFR4
SCHEMBL601169 0.67 SLC6A2 (0.37) SLC6A2NPC1
SCHEMBL17369262 0.66 SLC6A2 (0.35) SLC6A2NPC1FGFR4
SCHEMBL4874968 0.66 LRRK2 (0.42) SLC6A2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0417584-B1 N-substituted-4-pyrimidinamines and -pyrimidindiamines, a process for their preparation and their use as medicaments HOECHST MARION ROUSSEL INC (US) 1998-02-04 EP claimed
US-4983608-A Analgesics, cognition activators HOECHST-ROUSSELL PHARMACEUTICALS, INC. (US) 1991-01-08 US claimed
EP-0417584-B1 N-substituted-4-pyrimidinamines and -pyrimidindiamines, a process for their preparation and their use as medicaments HOECHST MARION ROUSSEL INC (US) 1998-02-04 EP disclosed
US-5179204-A Learning enhancement, analgesics HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1993-01-12 US disclosed
EP-0417584-A2 N-substituted-4-pyrimidinamines and -pyrimidindiamines, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1991-03-20 EP disclosed
US-4983608-A Analgesics, cognition activators HOECHST-ROUSSELL PHARMACEUTICALS, INC. (US) 1991-01-08 US disclosed