SCHEMBL8538715

SCHEMBL8538715

NC1=NC2(CS1)c1cc(-c3cncnc3)ccc1CC1CC(O)CCC12

nearest known ligand 0.46

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.46
CTSB P07858 2/20 0.46
CTSD P07339 6/20 0.41
BACE2 Q9Y5Z0 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8538718 1.00 BACE1 (0.46) BACE1CTSBCTSDBACE2
SCHEMBL9932194 0.87 BACE1 (0.47) BACE1CTSBCTSDBACE2
SCHEMBL9932066 0.82 BACE1 (0.44) BACE1CTSBCTSDBACE2
SCHEMBL10238054 0.81 BACE1 (0.56) BACE1CTSBCTSD
SCHEMBL9882480 0.81 BACE1 (0.56) BACE1CTSBCTSD
SCHEMBL9931896 0.81 BACE1 (0.56) BACE1CTSBCTSD
SCHEMBL9931899 0.81 BACE1 (0.56) BACE1CTSBCTSD
SCHEMBL9882441 0.81 BACE1 (0.56) BACE1CTSBCTSD
SCHEMBL8537151 0.80 BACE1 (0.55) BACE1CTSBCTSD
SCHEMBL8532624 0.80 BACE1 (0.55) BACE1CTSBCTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012071458-A1 HETEROCYCLIC INHIBITORS OF BETA - SECRETASE FOR THE TREATMENT OF NEURODEGENERATIVE DISEASES ARRAY BIOPHARMA INC. (US) 2012-05-31 WO disclosed