SCHEMBL854019

SCHEMBL854019

CC(C)(C)N(CCCOc1c(-c2ccccc2)[nH]c(=O)c2cc(F)ccc12)C(=O)O

nearest known ligand 0.56

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 17/20 0.56
PARP3 Q9Y6F1 10/20 0.54
PARP2 Q9UGN5 6/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL854082 0.81 PARP1 (0.64) PARP1PARP3PARP2
SCHEMBL854699 0.81 PARP1 (0.69) PARP1PARP3PARP2
Trifluoroacetic Acid SCHEMBL854159 0.80 PARP1 (0.55) PARP1PARP3PARP2
SCHEMBL854836 0.80 PARP1 (0.61) PARP1PARP3PARP2
SCHEMBL854607 0.79 PARP1 (0.76) PARP1PARP3PARP2
SCHEMBL854229 0.79 PARP1 (0.69) PARP1PARP3PARP2
SCHEMBL3713263 0.79 PARP1 (0.60) PARP1PARP3PARP2
Hydrochloric Acid SCHEMBL855640 0.78 PARP1 (0.74) PARP1PARP3PARP2
SCHEMBL853576 0.78 PARP1 (0.55) PARP1PARP3PARP2
SCHEMBL854579 0.78 PARP1 (0.86) PARP1PARP3PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2432765-A1 ISOQUINOLIN-1 (2H) -ONE DERIVATIVES AS PARP-1 INHIBITORS Nerviano Medical Sciences S.r.l. (IT) 2012-03-28 EP disclosed