SCHEMBL8540948

SCHEMBL8540948

O=C(O)c1c(-c2ccccc2)c2cc(OCc3ccccc3)ccc2n1Cc1cc2c(cc1Cl)OCO2

nearest known ligand 0.72

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 18/20 0.72
EDNRB P24530 17/20 0.72
S1PR1 P21453 1/20 0.47
PRKX P51817 1/20 0.47
ACVR1 Q04771 1/20 0.47
S1PR5 Q9H228 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8856895 0.95 EDNRB (0.71) EDNRAEDNRB
SCHEMBL8590639 0.95 EDNRA (0.64) EDNRAEDNRB
SCHEMBL8856638 0.94 EDNRA (0.78) EDNRAEDNRB
SCHEMBL8856815 0.94 EDNRB (0.74) EDNRAEDNRB
SCHEMBL8856820 0.94 EDNRA (0.66) EDNRAEDNRB
SCHEMBL8856631 0.92 EDNRB (0.65) EDNRAEDNRB
SCHEMBL8856822 0.92 EDNRA (0.70) EDNRAEDNRB
SCHEMBL8856577 0.92 EDNRB (0.64) EDNRAEDNRBS1PR1S1PR5
SCHEMBL8856755 0.92 EDNRB (0.65) EDNRAEDNRB
SCHEMBL8857076 0.92 EDNRB (0.64) EDNRAEDNRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0800389-A4 NOVEL COMPOUNDS SMITHKLINE BEECHAM CORP (US) 1998-04-29 EP disclosed
US-5684032-A ANTIINFLAMMATORY AGENTS, ANTIARTHRITIC, ANTIASTHMATIC AGENTS AND RESPIRATORY DISORDERS SMITHKLINE BEECHAM CORPORATION (US) 1997-11-04 US disclosed
EP-0800389-A1 NOVEL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1997-10-15 EP disclosed
WO-1996018393-A1 NOVEL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1996-06-20 WO disclosed