SCHEMBL8543715

SCHEMBL8543715

COc1ccc(N2CCN(C(=O)C3(C)CCc4c(C)c(O)c(C)c(C)c4O3)CC2)cc1

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.51
PTGS2 P35354 1/20 0.51
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
TSHR P16473 1/20 0.51
HTT P42858 1/20 0.50
ALDH1A1 P00352 2/20 0.46
BCHE P06276 7/20 0.45
ACHE P22303 7/20 0.45
AKR1C3 P42330 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.42
LMNA P02545 1/20 0.42
POLB P06746 1/20 0.42
MAPT P10636 1/20 0.42
PKM P14618 1/20 0.42
RAB9A P51151 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9266621 0.88 CYP3A4 (0.46) PTGS1PTGS2CYP1A2CYP3A4TSHR
SCHEMBL9690307 0.88 PTGS1 (0.53) PTGS1PTGS2CYP1A2CYP3A4TSHR
SCHEMBL8545535 0.85 HTT (0.45) HTTALDH1A1AKR1C3L3MBTL1KMT2A
SCHEMBL4309982 0.85 CYP3A4 (0.49) PTGS1PTGS2CYP1A2CYP3A4TSHR
SCHEMBL9690157 0.83 TSHR (0.49) PTGS1PTGS2CYP1A2CYP3A4TSHR
SCHEMBL4322635 0.82 GFER (0.42) PTGS1PTGS2CYP1A2CYP3A4TSHR
SCHEMBL4316353 0.82 PTGS1 (0.47) PTGS1PTGS2CYP1A2CYP3A4TSHR
SCHEMBL9690175 0.82 TSHR (0.50) PTGS1PTGS2CYP1A2CYP3A4TSHR
SCHEMBL4322552 0.80 MAPT (0.47) HTTALDH1A1AKR1C3KMT2AMEN1
SCHEMBL2059305 0.80 PTGS1 (0.64) PTGS1PTGS2CYP1A2CYP3A4TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0487510-A1 Pharmaceutically active amines THE UPJOHN COMPANY (US) 1992-05-27 EP claimed
EP-0358676-A1 PHARMACEUTICALLY ACTIVE AMINES THE UPJOHN COMPANY (US) 1990-03-21 EP claimed
EP-0293078-A1 Pharmaceutically active amines THE UPJOHN COMPANY (US) 1988-11-30 EP claimed
WO-1988008424-A1 PHARMACEUTICALLY ACTIVE AMINES THE UPJOHN COMPANY (US) 1988-11-03 WO claimed
EP-0587499-B1 Benzopyran compounds, process for their preparation and their use as cell protectors ADIR (FR) 1998-04-29 EP disclosed
US-5395834-A Antiarthritic agents or cardiovascular disorders ADIR ET COMPAGNIE (FR) 1995-03-07 US disclosed
US-5393775-A Administering a (2-chromanyl)alkylcarboxylic acid for disorders connected with peroxidation processes ADIR ET COMPAGNIE (FR) 1995-02-28 US disclosed
EP-0587499-A1 Benzopyran compounds, process for their preparation and their use as cell protectors ADIR ET COMPAGNIE (FR) 1994-03-16 EP disclosed
EP-0358676-A1 PHARMACEUTICALLY ACTIVE AMINES THE UPJOHN COMPANY (US) 1990-03-21 EP disclosed
WO-1988008424-A1 PHARMACEUTICALLY ACTIVE AMINES THE UPJOHN COMPANY (US) 1988-11-03 WO disclosed