SCHEMBL8546304

SCHEMBL8546304

CC(=CCCl)c1cccc(OCc2nc(-c3ccccc3)oc2C)c1

nearest known ligand 0.62

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KDR P35968 1/20 0.62
PTPN1 P18031 3/20 0.56
MAPT P10636 3/20 0.50
FFAR1 O14842 1/20 0.50
PPARG P37231 4/20 0.48
PPARA Q07869 4/20 0.48
TP53 P04637 2/20 0.47
POLB P06746 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8546298 1.00 KDR (0.62) KDRPTPN1MAPTFFAR1PPARG
SCHEMBL8546300 1.00 KDR (0.62) KDRPTPN1MAPTFFAR1PPARG
SCHEMBL8546210 0.91 KDR (0.67) KDRPTPN1MAPTFFAR1PPARG
SCHEMBL8546212 0.91 KDR (0.67) KDRPTPN1MAPTFFAR1PPARG
SCHEMBL9078622 0.89 PTPN1 (0.60) KDRPTPN1PPARGPPARA
SCHEMBL9078616 0.89 PTPN1 (0.60) KDRPTPN1PPARGPPARA
SCHEMBL9078620 0.89 PTPN1 (0.60) KDRPTPN1PPARGPPARA
SCHEMBL8547074 0.84 KDR (0.69) KDRMAPTFFAR1PPARGPPARA
SCHEMBL8546414 0.83 KDR (0.62) KDRPTPN1MAPTFFAR1PPARG
SCHEMBL9170685 0.83 KDR (0.62) KDRPTPN1MAPTFFAR1PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0759919-B1 AZOLIDINEDIONES AS ANTIHYPERGLYCEMIC AGENTS AMERICAN HOME PROD (US) 1998-11-11 EP disclosed
CN-1152312-A Novel pyrrolidinediones as antihyperglycemic agents AMERICAN HOME PROD (US) 1997-06-18 CN disclosed
EP-0759919-A1 NEW AZOLIDINEDIONES AS ANTIHYPERGLYCEMIC AGENTS AMERICAN HOME PRODUCTS CORPORATION (US) 1997-03-05 EP disclosed
US-5532256-A ORALLY ADMINISTERED ANTIDIABETIC AGENTS AMERICAN HOME PRODUCTS CORPORATION (US) 1996-07-02 US disclosed
US-5510360-A ADMINISTERING ORALLY, SIDE EFFECT REDUCTION AMERICAN HOME PRODUCTS CORPORATION (US) 1996-04-23 US disclosed
WO-1995031454-A1 NEW AZOLIDINEDIONES AS ANTIHYPERGLYCEMIC AGENTS AMERICAN HOME PRODUCTS CORPORATION (US) 1995-11-23 WO disclosed
US-5468762-A Antidiabetic agents for administering by mouth AMERICAN HOME PRODUCTS CORPORATION (US) 1995-11-21 US disclosed