SCHEMBL8549596

SCHEMBL8549596

COc1ccccc1-c1c(C(=O)O)n(Cc2ccc3nsnc3c2)c2ccc(N)cc12

nearest known ligand 0.57

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
EDNRB P24530 12/20 0.57
EDNRA P25101 9/20 0.57
CCR2 P41597 2/20 0.41
PTGES2 Q9H7Z7 1/20 0.38
PLA2G2A P14555 1/20 0.38
ABCB11 O95342 1/20 0.38
PTGES O14684 1/20 0.38
SERPINE1 P05121 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8548412 0.90 EDNRB (0.62) EDNRBEDNRAPLA2G2A
SCHEMBL8549602 0.88 EDNRB (0.46) EDNRBEDNRACCR2PTGES2PLA2G2A
SCHEMBL8546347 0.88 EDNRB (0.66) EDNRBEDNRASERPINE1
SCHEMBL8548299 0.86 EDNRB (0.54) EDNRBEDNRACCR2SERPINE1
SCHEMBL8553149 0.86 EDNRB (0.52) EDNRBEDNRACCR2PTGES2ABCB11
SCHEMBL8550267 0.85 EDNRB (0.77) EDNRBEDNRASERPINE1
SCHEMBL8552318 0.84 EDNRB (0.55) EDNRBEDNRACCR2SERPINE1
SCHEMBL8548047 0.83 EDNRB (0.43) EDNRBEDNRAPTGES2PLA2G2APTGES
SCHEMBL8624241 0.83 EDNRB (0.52) EDNRBEDNRACCR2
SCHEMBL8550371 0.82 EDNRB (0.53) EDNRBEDNRASERPINE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863898-A1 ENDOTHELIN RECEPTOR ANTAGONISTS MERCK PATENT GmbH (DE) 1998-09-16 EP disclosed
WO-1997019077-A1 ENDOTHELIN RECEPTOR ANTAGONISTS MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1997-05-29 WO disclosed