SCHEMBL8550158

SCHEMBL8550158

COc1ccc(N2CCN(CC[C@H]3OCCc4cc(C(N)=O)ccc43)CC2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 13/20 1.00
DRD2 P14416 8/20 1.00
HTR2A P28223 6/20 1.00
HTR1A P08908 6/20 1.00
DRD4 P21917 5/20 1.00
HTR1B P28222 5/20 0.82
SLC6A4 P31645 3/20 0.72
CA12 O43570 1/20 0.52
CA1 P00915 1/20 0.52
CA2 P00918 1/20 0.52
CA4 P22748 1/20 0.52
CA6 P23280 1/20 0.52
CA5A P35218 1/20 0.52
CA7 P43166 1/20 0.52
CA9 Q16790 1/20 0.52
CA13 Q8N1Q1 1/20 0.52
CA14 Q9ULX7 1/20 0.52
CA5B Q9Y2D0 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8550714 1.00 HTR1D (1.00) HTR1DDRD2HTR2AHTR1ADRD4
SCHEMBL7403625 1.00 HTR1D (1.00) HTR1DDRD2HTR2AHTR1ADRD4
SCHEMBL8549600 0.93 HTR1D (0.86) HTR1DDRD2HTR2AHTR1ADRD4
SCHEMBL7402753 0.93 HTR1D (0.86) HTR1DDRD2HTR2AHTR1ADRD4
SCHEMBL8551125 0.93 HTR1D (0.86) HTR1DDRD2HTR2AHTR1ADRD4
SCHEMBL5595821 0.90 HTR1D (1.00) HTR1DDRD2HTR2AHTR1ADRD4
SCHEMBL7401976 0.90 HTR1D (1.00) HTR1DDRD2HTR2AHTR1ADRD4
SCHEMBL8549606 0.90 HTR1D (1.00) HTR1DDRD2HTR2AHTR1ADRD4
SCHEMBL30628146 0.90 HTR1D (1.00) HTR1DDRD2HTR2AHTR1ADRD4
SCHEMBL7403048 0.90 HTR1D (0.82) HTR1DDRD2HTR2AHTR1ADRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0836599-A1 1,6-DISUBSTITUTED ISOCHROMANS FOR TREATMENT OF MIGRAINE HEADACHES PHARMACIA & UPJOHN COMPANY (US) 1998-04-22 EP claimed
WO-1997002259-A1 1,6-DISUBSTITUTED ISOCHROMANS FOR TREATMENT OF MIGRAINE HEADACHES PHARMACIA & UPJOHN COMPANY (US) 1997-01-23 WO claimed
EP-0836599-A1 1,6-DISUBSTITUTED ISOCHROMANS FOR TREATMENT OF MIGRAINE HEADACHES PHARMACIA & UPJOHN COMPANY (US) 1998-04-22 EP disclosed
WO-1997002259-A1 1,6-DISUBSTITUTED ISOCHROMANS FOR TREATMENT OF MIGRAINE HEADACHES PHARMACIA & UPJOHN COMPANY (US) 1997-01-23 WO disclosed