SCHEMBL8550185

SCHEMBL8550185

CC(=O)c1ccc(OCCc2nc(-c3ccccc3)oc2C)cc1

nearest known ligand 0.77

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PPARG P37231 19/20 0.77
PPARA Q07869 17/20 0.77
PPARD Q03181 6/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1122908 0.92 PPARG (0.78) PPARGPPARAPPARD
SCHEMBL12618028 0.89 PPARG (0.75) PPARGPPARAPPARD
SCHEMBL6959523 0.89 FFAR1 (0.70) PPARGPPARA
SCHEMBL1123237 0.88 PPARG (0.73) PPARGPPARAPPARD
SCHEMBL13721507 0.87 PPARG (0.65) PPARGPPARA
SCHEMBL4389208 0.87 PPARG (0.79) PPARGPPARAPPARD
SCHEMBL5110945 0.87 PPARG (1.00) PPARGPPARAPPARD
SCHEMBL3283978 0.86 PPARG (0.77) PPARGPPARAPPARD
SCHEMBL6381921 0.86 PPARA (0.70) PPARGPPARAPPARD
SCHEMBL5098728 0.85 PPARG (0.76) PPARGPPARAPPARD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7279485-B2 Substituted heterocyclic derivatives useful as antidiabetic and antiobesity agents and method BRISTOL-MYERS SQUIBB COMPANY (US) 2007-10-09 US disclosed
EP-0759919-B1 AZOLIDINEDIONES AS ANTIHYPERGLYCEMIC AGENTS AMERICAN HOME PROD (US) 1998-11-11 EP disclosed
EP-0759919-A1 NEW AZOLIDINEDIONES AS ANTIHYPERGLYCEMIC AGENTS AMERICAN HOME PRODUCTS CORPORATION (US) 1997-03-05 EP disclosed
US-5532256-A ORALLY ADMINISTERED ANTIDIABETIC AGENTS AMERICAN HOME PRODUCTS CORPORATION (US) 1996-07-02 US disclosed
WO-1995031454-A1 NEW AZOLIDINEDIONES AS ANTIHYPERGLYCEMIC AGENTS AMERICAN HOME PRODUCTS CORPORATION (US) 1995-11-23 WO disclosed
US-5468762-A Antidiabetic agents for administering by mouth AMERICAN HOME PRODUCTS CORPORATION (US) 1995-11-21 US disclosed