SCHEMBL8550993

SCHEMBL8550993

Cc1ccc(Cn2c(=O)n(CCN3CCC(C(=O)c4ccc(F)cc4)CC3)c3ccccc32)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 7/20 0.55
HTR2C P28335 4/20 0.55
HTR7 P34969 3/20 0.55
HTR6 P50406 3/20 0.55
KCNH2 Q12809 2/20 0.53
CYP3A4 P08684 4/20 0.53
CYP1A2 P05177 3/20 0.53
CYP2C9 P11712 3/20 0.53
ALDH1A1 P00352 2/20 0.53
HTR1A P08908 2/20 0.53
DRD2 P14416 2/20 0.53
HPGD P15428 2/20 0.53
MEN1 O00255 1/20 0.53
LMNA P02545 1/20 0.53
MAPT P10636 1/20 0.53
ADRA2B P18089 1/20 0.53
ADRA2C P18825 1/20 0.53
DRD1 P21728 1/20 0.53
DRD4 P21917 1/20 0.53
HTR1D P28221 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8019192 0.99 HTR2A (0.54) HTR2AHTR2CHTR7HTR6KCNH2
Hydrochloric Acid SCHEMBL8025211 0.94 HTR2A (0.60) HTR2AHTR2CHTR7HTR6KCNH2
Hydrochloric Acid SCHEMBL8021166 0.91 HTR2A (0.61) HTR2AHTR2CHTR7HTR6KCNH2
Hydrochloric Acid SCHEMBL8023021 0.90 HTR2A (0.55) HTR2AHTR2CHTR7HTR6KCNH2
Hydrochloric Acid SCHEMBL8023102 0.90 HTR2A (0.66) HTR2AHTR2CHTR7HTR6KCNH2
Hydrochloric Acid SCHEMBL8008723 0.90 HTR2A (0.54) HTR2AHTR2CHTR7HTR6KCNH2
Hydrochloric Acid SCHEMBL8020904 0.90 HTR2A (0.54) HTR2AHTR2CHTR7HTR6KCNH2
Hydrochloric Acid SCHEMBL8021159 0.89 HTR2A (0.52) HTR2AHTR2CHTR7HTR6KCNH2
Hydrochloric Acid SCHEMBL8023096 0.89 HRH1 (0.61) HTR2AHTR2CHTR7HTR6KCNH2
Dimethylamine SCHEMBL8023031 0.89 HTR2A (0.52) HTR2AHTR2CHTR7HTR6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0816356-A1 1-(2-(1-piperidinyl)-1-ethyl)-1,3-dihydro-2H-benzimidazole derivatives and their pharmaceutical use ELI LILLY AND COMPANY LIMITED (GB) 1998-01-07 EP disclosed