SCHEMBL8551064

SCHEMBL8551064

CCCCS(=O)(=O)Nc1ccc2c(c1)c(-c1ccc(OC)cc1OC)c(OC(=O)O)n2Cc1ccc2nsnc2c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EDNRB P24530 6/20 0.47
EDNRA P25101 2/20 0.40
CA2 P00918 1/20 0.37
CA9 Q16790 1/20 0.37
KDM4E B2RXH2 2/20 0.36
HSD17B10 Q99714 2/20 0.36
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
MAPT P10636 4/20 0.35
CYP17A1 P05093 1/20 0.34
KIT P10721 1/20 0.34
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
MEN1 O00255 1/20 0.34
GAA P10253 1/20 0.34
KMT2A Q03164 1/20 0.34
POLB P06746 1/20 0.34
MAP2K4 P45985 1/20 0.34
JAK1 P23458 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8550374 0.92 EDNRB (0.43) EDNRBEDNRACA9KDM4EHSD17B10
SCHEMBL8551061 0.90 EDNRB (0.57) EDNRBEDNRACA2CA9KDM4E
SCHEMBL8548080 0.90 EDNRB (0.49) EDNRBEDNRACA2CA9KDM4E
SCHEMBL8546571 0.89 EDNRB (0.47) EDNRBEDNRACA9KDM4EHSD17B10
SCHEMBL8550229 0.86 EDNRB (0.48) EDNRBEDNRACA2CA9KDM4E
SCHEMBL8551085 0.85 EDNRB (0.45) EDNRBEDNRACA2CA9KDM4E
SCHEMBL8548088 0.85 EDNRB (0.47) EDNRBEDNRAKDM4EHSD17B10ALDH1A1
SCHEMBL8550960 0.84 EDNRB (0.66) EDNRBEDNRAKDM4EMAPTMEN1
SCHEMBL8551203 0.83 EDNRB (0.52) EDNRBEDNRAKDM4EHSD17B10ALDH1A1
SCHEMBL8551102 0.83 EDNRB (0.45) EDNRBEDNRAKDM4EHSD17B10ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863898-A1 ENDOTHELIN RECEPTOR ANTAGONISTS MERCK PATENT GmbH (DE) 1998-09-16 EP disclosed
WO-1997019077-A1 ENDOTHELIN RECEPTOR ANTAGONISTS MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1997-05-29 WO disclosed