SCHEMBL8551100

SCHEMBL8551100

CCCCS(=O)(=O)Nc1ccc2c(c1)c(-c1ccc(C=O)cc1)c(C(=O)O)n2Cc1ccc2nsnc2c1

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
EDNRB P24530 11/20 0.56
EDNRA P25101 8/20 0.50
SERPINE1 P05121 5/20 0.49
HPGD P15428 3/20 0.40
ALDH1A1 P00352 2/20 0.40
KDM4E B2RXH2 1/20 0.40
HSD17B10 Q99714 1/20 0.40
LMNA P02545 3/20 0.36
MEN1 O00255 1/20 0.36
HTT P42858 1/20 0.36
KMT2A Q03164 1/20 0.36
PSMD14 O00487 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8548086 0.92 EDNRB (0.58) EDNRBEDNRASERPINE1HPGDALDH1A1
SCHEMBL8551102 0.89 EDNRB (0.45) EDNRBEDNRASERPINE1HPGDALDH1A1
SCHEMBL8551723 0.89 EDNRB (0.58) EDNRBEDNRASERPINE1
SCHEMBL8546569 0.87 EDNRB (0.59) EDNRBEDNRASERPINE1HPGDALDH1A1
SCHEMBL8546719 0.86 EDNRB (0.69) EDNRBEDNRASERPINE1
SCHEMBL8548322 0.86 EDNRB (0.42) EDNRBEDNRASERPINE1HPGDALDH1A1
SCHEMBL8548900 0.84 EDNRB (0.53) EDNRBEDNRASERPINE1LMNAPSMD14
SCHEMBL8550371 0.83 EDNRB (0.53) EDNRBEDNRASERPINE1HPGDALDH1A1
SCHEMBL8551061 0.82 EDNRB (0.57) EDNRBEDNRASERPINE1HPGDALDH1A1
SCHEMBL8550747 0.81 EDNRB (0.58) EDNRBEDNRASERPINE1LMNAPSMD14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863898-A1 ENDOTHELIN RECEPTOR ANTAGONISTS MERCK PATENT GmbH (DE) 1998-09-16 EP disclosed
WO-1997019077-A1 ENDOTHELIN RECEPTOR ANTAGONISTS MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1997-05-29 WO disclosed