SCHEMBL8551285

SCHEMBL8551285

Cc1ccccc1-c1n[nH]c(=O)c2c(Br)cccc12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 2/20 0.42
CHEK1 O14757 2/20 0.41
LMNA P02545 2/20 0.40
TSHR P16473 2/20 0.40
ATM Q13315 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
NOTUM Q6P988 1/20 0.39
PRMT5 O14744 1/20 0.39
WDR77 Q9BQA1 1/20 0.39
MAPK1 P28482 2/20 0.38
S1PR2 O95136 1/20 0.38
TP53 P04637 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
HTR7 P34969 1/20 0.38
ROCK1 Q13464 3/20 0.37
PDE7A Q13946 2/20 0.37
NPC1 O15118 2/20 0.37
RAB9A P51151 1/20 0.37
DCUN1D1 Q96GG9 1/20 0.36
KDM4E B2RXH2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8548318 0.88 AR (0.46) ARCHEK1LMNATSHRATM
SCHEMBL8547990 0.83 NPSR1 (0.50) CHEK1LMNATSHRATMNPSR1
SCHEMBL8552195 0.83 AR (0.42) ARCHEK1LMNATSHRATM
SCHEMBL8549626 0.83 AR (0.42) ARCHEK1LMNATSHRATM
SCHEMBL8546629 0.83 PARP1 (0.40) LMNATSHRMAPK1S1PR2TP53
SCHEMBL8548460 0.81 NPSR1 (0.62) ATMNPSR1MAPK1TP53ROCK1
SCHEMBL8547999 0.80 NOTUM (0.43) ARATMNPSR1NOTUMROCK2
SCHEMBL30108722 0.76 PDE4A (0.43) ARLMNATSHRMAPK1S1PR2
SCHEMBL28934651 0.76 PDE4A (0.43) ARLMNATSHRMAPK1S1PR2
SCHEMBL15031985 0.75 PRMT5 (0.53) ARLMNATSHRATMNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825187-A1 Condensed pyridazinyl guanidines, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-25 EP disclosed