SCHEMBL8551626

SCHEMBL8551626

CCOC(=O)Oc1c(-c2ccc(OC)cc2OC)c2cc(NC(=O)OC)ccc2n1Cc1ccc2nsnc2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EDNRB P24530 6/20 0.46
MAPT P10636 10/20 0.40
EDNRA P25101 2/20 0.40
NPC1 O15118 4/20 0.39
RAB9A P51151 4/20 0.39
MEN1 O00255 4/20 0.39
KMT2A Q03164 4/20 0.39
SMN1; SMN2 Q16637 4/20 0.39
GAA P10253 3/20 0.39
POLB P06746 2/20 0.38
HTT P42858 1/20 0.37
LMNA P02545 1/20 0.37
KDM4E B2RXH2 3/20 0.37
HSD17B10 Q99714 2/20 0.37
TSHR P16473 1/20 0.37
ATM Q13315 1/20 0.37
TP53 P04637 1/20 0.36
CA2 P00918 1/20 0.36
CA9 Q16790 1/20 0.36
HPGD P15428 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8548161 0.95 EDNRB (0.46) EDNRBMAPTEDNRANPC1RAB9A
SCHEMBL8545641 0.91 EDNRB (0.42) EDNRBMAPTEDNRANPC1RAB9A
SCHEMBL8550229 0.91 EDNRB (0.48) EDNRBMAPTEDNRANPC1RAB9A
SCHEMBL8553017 0.90 EDNRB (0.54) EDNRBMAPTEDNRANPC1RAB9A
SCHEMBL8547254 0.88 EDNRB (0.46) EDNRBMAPTEDNRARAB9AMEN1
SCHEMBL8547971 0.88 EDNRB (0.48) EDNRBMAPTEDNRAMEN1KMT2A
SCHEMBL8547424 0.87 EDNRB (0.61) EDNRBMAPTEDNRAMEN1KMT2A
SCHEMBL8547270 0.86 EDNRB (0.42) EDNRBMAPTEDNRANPC1RAB9A
SCHEMBL8548911 0.85 EDNRB (0.46) EDNRBMAPTEDNRASMN1; SMN2GAA
SCHEMBL8549274 0.85 EDNRB (0.55) EDNRBMAPTEDNRANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863898-A1 ENDOTHELIN RECEPTOR ANTAGONISTS MERCK PATENT GmbH (DE) 1998-09-16 EP disclosed
WO-1997019077-A1 ENDOTHELIN RECEPTOR ANTAGONISTS MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1997-05-29 WO disclosed