SCHEMBL8552546

SCHEMBL8552546

CCOC(=O)c1cccc(N(C(N)=O)c2ccc(Oc3ccnc4cc(OC)c(OC)cc34)cc2)c1

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDR P35968 8/20 0.50
AURKA O14965 2/20 0.50
LCK P06239 2/20 0.50
MET P08581 2/20 0.50
TEK Q02763 2/20 0.50
AURKB Q96GD4 2/20 0.50
ABL1 P00519 1/20 0.50
LYN P07948 1/20 0.50
PDGFRA P16234 9/20 0.49
FGFR2 P21802 1/20 0.48
PDGFRB P09619 1/20 0.47
KIT P10721 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8556378 0.85 PDGFRA (0.61) KDRAURKALCKMETTEK
SCHEMBL8554460 0.84 KDR (0.62) KDRAURKALCKMETTEK
SCHEMBL8556873 0.84 PDGFRA (0.62) KDRAURKALCKMETTEK
SCHEMBL22972011 0.83 EGFR (0.60) KDRAURKALCKMETTEK
SCHEMBL8554907 0.83 KDR (0.55) KDRAURKALCKMETTEK
SCHEMBL8552489 0.83 PDGFRA (0.65) KDRAURKALCKMETTEK
SCHEMBL8553956 0.81 FGFR2 (0.59) KDRAURKALCKMETTEK
SCHEMBL8551461 0.81 PDGFRA (0.59) KDRAURKALCKMETTEK
SCHEMBL8554250 0.81 PDGFRA (0.64) KDRAURKALCKMETTEK
SCHEMBL24724228 0.81 EGFR (0.56) KDRAURKALCKMETTEK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0860433-A1 QUINOLINE DERIVATIVES AND QUINAZOLINE DERIVATIVES INHIBITING AUTOPHOSPHORYLATION OF GROWTH FACTOR RECEPTOR ORIGINATING IN PLATELET AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME KIRIN BEER KABUSHIKI KAISHA (JP) 1998-08-26 EP disclosed