SCHEMBL8554659

SCHEMBL8554659

CS(=O)(=O)CCC(CNC(=O)c1ccccc1)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.45
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
ITGAV P06756 4/20 0.43
GPR139 Q6DWJ6 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
S1PR2 O95136 1/20 0.41
S1PR4 O95977 1/20 0.41
S1PR3 Q99500 1/20 0.41
TACR2 P21452 2/20 0.41
SCN9A Q15858 1/20 0.41
SLC6A2 P23975 2/20 0.40
SLC6A4 P31645 2/20 0.40
SLC6A3 Q01959 2/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
MCHR1 Q99705 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8597116 0.85 NPC1 (0.54) NPC1RAB9AITGAVGPR139SMN1; SMN2
SCHEMBL8308087 0.85 NPC1 (0.43) NPC1RAB9AITGAVSMN1; SMN2SLC6A2
SCHEMBL6161768 0.84 NPC1 (0.49) HPGDNPC1RAB9AITGAVGPR139
SCHEMBL5866425 0.84 NPC1 (0.49) HPGDNPC1RAB9AITGAVGPR139
SCHEMBL7045680 0.81 TACR2 (0.47) HPGDNPC1RAB9AGPR139SMN1; SMN2
SCHEMBL5866364 0.81 TACR2 (0.47) HPGDNPC1RAB9AGPR139SMN1; SMN2
SCHEMBL6665274 0.81 SLC6A2 (0.48) HPGDNPC1RAB9AGPR139SMN1; SMN2
SCHEMBL6665281 0.81 SLC6A2 (0.48) HPGDNPC1RAB9AGPR139SMN1; SMN2
SCHEMBL4468917 0.79 SLC6A2 (0.50) SLC6A2SLC6A4SLC6A3CYP3A4CYP2D6
SCHEMBL6425161 0.79 TACR2 (0.65) TACR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0882038-A1 NOVEL SUBSTITUTED N-METHYL-N-(4-(PIPERIDIN-1-YL)-2-(ARYL)BUTYL)BENZAMIDES USEFUL FOR THE TREATMENT OF ALLERGIC DISEASES HOECHST MARION ROUSSEL, INC. (US) 1998-12-09 EP disclosed
WO-1997030990-A1 NOVEL SUBSTITUTED N-METHYL-N-(4-(PIPERIDIN-1-YL)-2-(ARYL)BUTYL)BENZAMIDES USEFUL FOR THE TREATMENT OF ALLERGIC DISEASES HOECHST MARION ROUSSEL, INC. (US) 1997-08-28 WO disclosed