SCHEMBL8559300

SCHEMBL8559300

CN(CC(O)c1ccc(Cl)c(Cl)c1)C(=O)OC(C)(C)C

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
F2R P25116 4/20 0.52
SLC6A2 P23975 2/20 0.41
SLC6A4 P31645 2/20 0.41
SLC6A3 Q01959 2/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
TACR2 P21452 1/20 0.36
AOC3 Q16853 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL756562 0.86 F2R (0.42) F2RSLC6A2SLC6A4SLC6A3CYP3A4
SCHEMBL4352299 0.85 AOC3 (0.53) F2RCYP3A4CYP2D6LMNASMN1; SMN2
SCHEMBL2528524 0.84 F2R (0.40) F2RSLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL8483223 0.84 TACR2 (0.41) F2RTACR2
SCHEMBL10878881 0.83 MAPT (0.44) SLC6A2CYP3A4CYP2D6ALDH1A1LMNA
SCHEMBL11212431 0.83 MAPT (0.44) SLC6A2CYP3A4CYP2D6ALDH1A1LMNA
SCHEMBL1690586 0.83 F2R (0.41) F2RSLC6A2SLC6A4SLC6A3CYP3A4
SCHEMBL4870085 0.83 TACR2 (0.46) TACR2
SCHEMBL1690588 0.83 F2R (0.41) F2RSLC6A2SLC6A4SLC6A3CYP3A4
SCHEMBL756561 0.83 TACR2 (0.46) TACR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5726313-A Substituted arylaliphatic compounds, method of preparing them and pharmaceutical compositions in which they are present SANOFI (FR) 1998-03-10 US disclosed
EP-0700386-A1 NEUROKININ RECEPTOR ANTAGONISTS SANOFI (FR) 1996-03-13 EP disclosed
WO-1995026338-A1 NEUROKININ RECEPTOR ANTAGONISTS SANOFI (FR) 1995-10-05 WO disclosed