SCHEMBL8559459

SCHEMBL8559459

Nc1cccc(Nc2ccc(C(F)(F)F)cc2[N+](=O)[O-])c1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 1/20 0.69
AKR1C4 P17516 1/20 0.69
AKR1C3 P42330 1/20 0.69
AKR1C2 P52895 1/20 0.69
AKR1C1 Q04828 1/20 0.69
MAPK1 P28482 6/20 0.63
EPAS1 Q99814 2/20 0.58
KIF11 P52732 1/20 0.50
FBP1 P09467 1/20 0.49
MAPT P10636 7/20 0.49
MEN1 O00255 3/20 0.48
KMT2A Q03164 3/20 0.48
KCNMA1 Q12791 1/20 0.48
ALDH1A1 P00352 3/20 0.48
GAA P10253 2/20 0.48
KDM4E B2RXH2 1/20 0.48
GFER P55789 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
ARNT P27540 1/20 0.47
RAB9A P51151 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8559386 0.91 AKR1B1 (0.77) AKR1B1AKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL2646781 0.86 AKR1B1 (0.70) AKR1B1AKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL10529983 0.85 MAPK1 (0.76) AKR1B1AKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL13811262 0.85 MAPK1 (0.75) AKR1B1AKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL11468688 0.85 AKR1B1 (0.72) AKR1B1AKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL2641949 0.85 AKR1B1 (0.69) AKR1B1AKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL1668253 0.85 AKR1B1 (0.69) AKR1B1AKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL11392520 0.82 MAPK1 (0.84) AKR1B1AKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL2493312 0.81 AKR1B1 (0.65) AKR1B1AKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL11515701 0.81 MAPT (0.72) MAPK1MAPTMEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0616807-B1 Benzimidazole useful in the treatment of central nervous system disorders NEUROSEARCH AS (DK) 1998-07-08 EP disclosed
US-4179436-A DYEING POLYESTERS BAYER AKTIENGESELLSCHAFT (DE) 1979-12-18 US disclosed
US-4163013-A Diphenylamine-azo-hydrocarbylsulfonylphenyl dyestuffs BAYER AKTIENGESELLSCHAFT (DE) 1979-07-31 US disclosed