SCHEMBL8559619

SCHEMBL8559619

Cc1cn2cccc(OCc3ccc(Br)cc3F)c2n1

nearest known ligand 0.58

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
PTGER1 P34995 6/20 0.41
MAPK14 Q16539 6/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10532132 0.84 GUCY1B2 (0.46)
SCHEMBL9747203 0.80 PSEN1 (0.43)
SCHEMBL12797510 0.79 HRH3 (0.48) PTGER1
SCHEMBL8565013 0.78 GUCY1B2 (0.47)
SCHEMBL8567556 0.78 PSEN1 (0.48)
SCHEMBL12797495 0.77 NPC1 (0.59) PTGER1
SCHEMBL2191140 0.77 MEN1 (0.51)
SCHEMBL9749030 0.77 PSEN1 (0.53)
SCHEMBL9748883 0.77 PTGER1 (0.44) PTGER1
SCHEMBL12848887 0.77 PPARG (0.48) PTGER1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0596406-B1 Imidazo (1,2-a) Pyridines as bradykinin antagonists FUJISAWA PHARMACEUTICAL CO (JP) 1998-12-16 EP disclosed
US-5750699-A HALOGENATING OF CORRESPONDING COMPOUND FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-05-12 US disclosed
US-5574042-A ANTAGONIST FOR BRADYKININS AS ANTIALLERGENS, AUTOIMMUNE DISEASES, ANTIINFLAMMATORY AGENTS, SHOCK OR PAIN FUJISAWA PHARMACEUTICAL CO., LTD (JP) 1996-11-12 US disclosed
EP-0596406-A1 Imidazo (1,2-a) Pyridines as bradykinin antagonists FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-05-11 EP disclosed