SCHEMBL8559971

SCHEMBL8559971

CS(=O)(=O)[N+]1(NC(=O)C(CCCc2ccccc2)NCc2ccccc2)CC2(CCNCC2)c2ccccc21

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 13/20 0.40
TLR2 O60603 2/20 0.34
ATM Q13315 1/20 0.31
TMPRSS2 O15393 1/20 0.31
TMPRSS11D O60235 1/20 0.31
F2 P00734 1/20 0.31
F10 P00742 1/20 0.31
PLG P00747 1/20 0.31
MMP3 P08254 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8559552 0.92 TACR1 (0.52) TACR1
SCHEMBL8558385 0.88 TACR1 (0.40) TACR1ATM
SCHEMBL8559103 0.87 TACR1 (0.51) TACR1
SCHEMBL8562658 0.86 TACR1 (0.47) TACR1
SCHEMBL8563510 0.82 TACR1 (0.44) TACR1
SCHEMBL8562925 0.82 TACR1 (0.51) TACR1
Hydrochloric Acid SCHEMBL8560263 0.81 TACR1 (0.50) TACR1
SCHEMBL8558359 0.81 TACR1 (0.51) TACR1
SCHEMBL8559375 0.81 TACR1 (0.51) TACR1
Hydrochloric Acid SCHEMBL8625895 0.81 TACR1 (0.43) TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5811431-A Spiro-substituted azacyclic derivatives and their use as therapeutic agents MERCK SHARP & DOHME LTD. (GB) 1998-09-22 US disclosed