SCHEMBL8560618

SCHEMBL8560618

Cc1cccc(C(=O)Nc2nc(C)cs2)c1

nearest known ligand 0.79

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GCK P35557 11/20 0.79
GRM5 P41594 1/20 0.76
NPC1 O15118 2/20 0.74
RAB9A P51151 2/20 0.74
HPGD P15428 1/20 0.72
SMN1; SMN2 Q16637 1/20 0.72
LMNA P02545 1/20 0.72
MAPT P10636 2/20 0.70
USP2 O75604 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7350718 0.86 GCK (0.72) GCKGRM5NPC1RAB9AHPGD
SCHEMBL21221226 0.86 GCK (0.72) GCKGRM5NPC1RAB9AHPGD
SCHEMBL1270190 0.85 NPC1 (1.00) GCKGRM5NPC1RAB9AHPGD
SCHEMBL3509220 0.85 NPC1 (0.75) GCKGRM5NPC1RAB9AHPGD
SCHEMBL19820469 0.84 GCK (0.69) GCKGRM5NPC1RAB9AHPGD
SCHEMBL19813926 0.84 GCK (0.69) GCKGRM5NPC1RAB9AHPGD
SCHEMBL14757305 0.83 GCK (0.73) GCKGRM5NPC1RAB9AHPGD
SCHEMBL2754003 0.83 SCD (0.69) NPC1RAB9AHPGDSMN1; SMN2LMNA
SCHEMBL4757037 0.83 GCK (0.58) GCKGRM5NPC1RAB9AHPGD
SCHEMBL1884815 0.82 MAPT (0.73) NPC1RAB9ASMN1; SMN2LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0815108-A1 CYCLIC UREA HIV PROTEASE INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1998-01-07 EP claimed
US-5683999-A Cyclic urea HIV protease inhibitors THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1997-11-04 US claimed
EP-0815108-A1 CYCLIC UREA HIV PROTEASE INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1998-01-07 EP disclosed
US-5683999-A Cyclic urea HIV protease inhibitors THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1997-11-04 US disclosed