SCHEMBL8560754

SCHEMBL8560754

C=CC(=O)OCCNS(=O)(=O)CCCCCCCC

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 7/20 0.54
HPGD P15428 1/20 0.54
ALDH1A1 P00352 3/20 0.46
CYP3A4 P08684 1/20 0.46
RELA Q04206 4/20 0.43
ZDHHC20 Q5W0Z9 1/20 0.41
ZDHHC2 Q9UIJ5 1/20 0.41
HCAR2 Q8TDS4 2/20 0.39
TP53 P04637 2/20 0.39
HIF1A Q16665 2/20 0.39
HSD17B10 Q99714 1/20 0.39
ATM Q13315 1/20 0.38
THRB P10828 1/20 0.37
EPHX2 P34913 1/20 0.37
CA2 P00918 2/20 0.36
CA12 O43570 1/20 0.36
CA7 P43166 1/20 0.36
CA9 Q16790 1/20 0.36
CA14 Q9ULX7 1/20 0.36
CA1 P00915 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29564360 1.00 TSHR (0.54) TSHRHPGDALDH1A1CYP3A4RELA
SCHEMBL11104966 0.86 TSHR (0.46) TSHRHPGDALDH1A1CYP3A4RELA
SCHEMBL9568651 0.83 TSHR (0.52) TSHRHPGDALDH1A1CYP3A4ZDHHC20
SCHEMBL10748682 0.83 TSHR (0.48) TSHRHPGDALDH1A1CYP3A4ZDHHC20
SCHEMBL10748508 0.81 TSHR (0.46) TSHRHPGDALDH1A1CYP3A4ZDHHC20
SCHEMBL8565012 0.80 TSHR (0.59) TSHRRELATHRBCA2CA12
SCHEMBL29107019 0.77 TSHR (0.62) TSHRHPGDALDH1A1CYP3A4ZDHHC20
SCHEMBL27517006 0.77 TSHR (0.58) TSHRHPGDALDH1A1CYP3A4HCAR2
SCHEMBL11828624 0.77 TSHR (0.62) TSHRHPGDALDH1A1CYP3A4ZDHHC20
SCHEMBL9442075 0.76 TSHR (0.84) TSHRHPGDALDH1A1CYP3A4HCAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5725789-A FOR FABRICS; POLYALKOXYLATED POLYURETHANE, FLUOROCHEMICAL ACRYLATE POLYMER MINNESOTA MINING AND MANUFACTURING COMPANY (US) 1998-03-10 US claimed
WO-1996030584-A1 AQUEOUS OIL AND WATER REPELLENT COMPOSITIONS MINNESOTA MINING AND MANUFACTURING COMPANY (US) 1996-10-03 WO claimed
CN-100347590-C Liquid crystal component KONINKL PHILIPS ELECTRONICS NV (NL) 2007-11-07 CN disclosed
CN-1732394-A Liquid crystal component KONINKL PHILIPS ELECTRONICS NV (NL) 2006-02-08 CN disclosed
US-5725789-A FOR FABRICS; POLYALKOXYLATED POLYURETHANE, FLUOROCHEMICAL ACRYLATE POLYMER MINNESOTA MINING AND MANUFACTURING COMPANY (US) 1998-03-10 US disclosed
WO-1996030584-A1 AQUEOUS OIL AND WATER REPELLENT COMPOSITIONS MINNESOTA MINING AND MANUFACTURING COMPANY (US) 1996-10-03 WO disclosed