SCHEMBL8562282

SCHEMBL8562282

CCOC(=O)C(C)CC1(c2ccccc2)CNC(=O)N1c1ccc2c(c1)CCN(C(=O)C(F)(F)F)CC2

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 3/20 0.35
ESR2 Q92731 3/20 0.35
TMEM97 Q5BJF2 8/20 0.34
SIGMAR1 Q99720 8/20 0.34
HTR1A P08908 1/20 0.34
CHRM5 P08912 1/20 0.34
SLC6A2 P23975 1/20 0.34
HRH2 P25021 1/20 0.34
ADRA1D P25100 1/20 0.34
HTR1B P28222 1/20 0.34
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34
HTR1E P28566 1/20 0.34
HRH1 P35367 1/20 0.34
HTR2B P41595 1/20 0.34
SLC6A3 Q01959 1/20 0.34
PDK2 Q15119 1/20 0.33
ALDH1A1 P00352 2/20 0.32
KDM4E B2RXH2 1/20 0.32
MTNR1B P49286 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8565993 0.78 ESR1 (0.40) ESR1ESR2ALDH1A1OPRM1TSHR
SCHEMBL8561377 0.75 ESR1 (0.41) ESR1ESR2TMEM97SIGMAR1ALDH1A1
SCHEMBL8560509 0.75 TMEM97 (0.42) TMEM97SIGMAR1HTR1ACHRM5SLC6A2
Hydrochloric Acid SCHEMBL8561493 0.74 TMEM97 (0.42) TMEM97SIGMAR1HTR1ACHRM5SLC6A2
SCHEMBL8561814 0.74 ESR1 (0.36) ESR1ESR2TMEM97SIGMAR1HTR1A
SCHEMBL8561816 0.72 ESR1 (0.36) ESR1ESR2TMEM97SIGMAR1HTR1A
SCHEMBL8895074 0.71 ESR1 (0.39) ESR1ESR2TMEM97SIGMAR1HTR1A
SCHEMBL8895079 0.71 ESR1 (0.39) ESR1ESR2TMEM97SIGMAR1HTR1A
SCHEMBL8565811 0.71 NOTUM (0.40) TMEM97SIGMAR1HTR1ACHRM5SLC6A2
SCHEMBL8562345 0.71 ESR1 (0.39) ESR1ESR2TMEM97SIGMAR1HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5827849-A HAVING INHIBITORY EFFECT ON INFLAMMATION AND BONE DEGRADATION, ANTITHROMBOTIC, ANTIAGGREGATORY AND TUMOR- OR METASTASIS-INHIBITING EFFECT KARL THOMAE GMBH (DE) 1998-10-27 US disclosed