SCHEMBL8563071

SCHEMBL8563071

COc1ccccc1CNC(COCc1ccccc1)C(=O)N[N+]1(S(C)(=O)=O)CC2(CCNCC2)c2ccccc21

nearest known ligand 0.52

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 19/20 0.52
ITGA4 P13612 1/20 0.37
ITGB7 P26010 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8565628 0.99 TACR1 (0.51) TACR1ITGA4ITGB7
SCHEMBL8562658 0.91 TACR1 (0.47) TACR1
SCHEMBL8563009 0.91 TACR1 (0.51) TACR1
SCHEMBL8557846 0.90 TACR1 (0.43) TACR1
SCHEMBL8563529 0.89 TACR1 (0.41) TACR1
SCHEMBL8565455 0.89 TACR1 (0.51) TACR1
SCHEMBL8558335 0.89 TACR1 (0.53) TACR1
SCHEMBL8563364 0.88 TACR1 (0.47) TACR1
Hydrochloric Acid SCHEMBL8566329 0.88 TACR1 (0.52) TACR1
SCHEMBL8564018 0.88 TACR1 (0.53) TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5811431-A Spiro-substituted azacyclic derivatives and their use as therapeutic agents MERCK SHARP & DOHME LTD. (GB) 1998-09-22 US disclosed