SCHEMBL8563078

SCHEMBL8563078

O=C1C(Br)CCN1c1ncccn1

nearest known ligand 0.39

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.39
CYP2C19 P33261 1/20 0.39
DRD2 P14416 2/20 0.37
HTR1A P08908 1/20 0.37
DRD4 P21917 1/20 0.37
CRBN Q96SW2 1/20 0.36
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8563081 1.00 KDM4E (0.39) KDM4ECYP2C19DRD2HTR1ADRD4
SCHEMBL7621523 0.80 CRBN (0.53) KDM4ECRBNALDH1A1
SCHEMBL7621521 0.80 CRBN (0.53) KDM4ECRBNALDH1A1
SCHEMBL7621516 0.80 CRBN (0.53) KDM4ECRBNALDH1A1
SCHEMBL8560932 0.76 GAA (0.37) CYP2C19ALDH1A1
SCHEMBL7614141 0.73 USP2 (0.44) KDM4EDRD2ALDH1A1
SCHEMBL7614145 0.73 USP2 (0.44) KDM4EDRD2ALDH1A1
SCHEMBL7624260 0.73 TDP1 (0.51) KDM4ECYP2C19ALDH1A1
SCHEMBL7620756 0.73 KDM4E (0.40) KDM4E
SCHEMBL7624265 0.73 TDP1 (0.51) KDM4ECYP2C19ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5804577-A ANTIBIOTICS HOFFMANN-LA ROCHE INC. (US) 1998-09-08 US disclosed
EP-0761673-A1 Cephalosporin derivatives F. HOFFMANN-LA ROCHE AG (CH) 1997-03-12 EP disclosed