SCHEMBL8563246

SCHEMBL8563246

COC(=O)CCC1(N2CCN(c3ccc4c(c3)CCN(C(=O)C(F)(F)F)CC4)C2=O)CCCCC1

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 3/20 0.39
ESR2 Q92731 3/20 0.39
BACE1 P56817 1/20 0.35
HDAC6 Q9UBN7 1/20 0.32
HRH3 Q9Y5N1 2/20 0.31
ABHD6 Q9BV23 1/20 0.31
TYRO3 Q06418 1/20 0.31
MERTK Q12866 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8559778 0.89 TP53 (0.36)
SCHEMBL8558361 0.85 ESR1 (0.40) ESR1ESR2HDAC6HRH3ABHD6
SCHEMBL8563649 0.80 TMEM97 (0.38) HRH3
SCHEMBL8561833 0.77 ESR1 (0.39) ESR1ESR2BACE1HDAC6HRH3
SCHEMBL8559203 0.76 ESR1 (0.38) ESR1ESR2BACE1HDAC6ABHD6
SCHEMBL8567428 0.75 ESR1 (0.40) ESR1ESR2HDAC6ABHD6TYRO3
SCHEMBL8567424 0.75 ESR1 (0.40) ESR1ESR2HDAC6ABHD6TYRO3
SCHEMBL8568710 0.74 F10 (0.39) ESR1ESR2
SCHEMBL8568715 0.74 F10 (0.39) ESR1ESR2
SCHEMBL8562059 0.73 ESR1 (0.36) ESR1ESR2BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5827849-A HAVING INHIBITORY EFFECT ON INFLAMMATION AND BONE DEGRADATION, ANTITHROMBOTIC, ANTIAGGREGATORY AND TUMOR- OR METASTASIS-INHIBITING EFFECT KARL THOMAE GMBH (DE) 1998-10-27 US disclosed